Restricted collision coupling of the adenosine A2Areceptor is due to its agonist-induced confinement in the membrane

被引:0
|
作者
Patrick Thurner
Simon Keuerleber
Ingrid Gsandtner
Christoph Gruber
Michael Freissmuth
Jürgen Zezula
机构
[1] Medical University of Vienna,Institute of Pharmacology, Center for Physiology and Pharmacology
关键词
Caffeine; Adenosine Receptor; Radioligand Binding; Docking Site; Diffusion Mode;
D O I
10.1186/2050-6511-13-S1-A81
中图分类号
学科分类号
摘要
引用
收藏
相关论文
共 50 条
  • [31] N-terminal and C-terminal plasma membrane anchoring modulate differently agonist-induced activation of cytosolic phospholipase A2
    Klapisz, E
    Ziari, M
    Wendum, D
    Koumanov, K
    Brachet-Ducos, C
    Olivier, JL
    Béréziat, G
    Trugnan, G
    Masliah, J
    EUROPEAN JOURNAL OF BIOCHEMISTRY, 1999, 265 (03): : 957 - 966
  • [32] CYCLIC-AMP ENHANCES AGONIST-INDUCED CA2+ ENTRY INTO ENDOTHELIAL-CELLS BY ACTIVATION OF POTASSIUM CHANNELS AND MEMBRANE HYPERPOLARIZATION
    GRAIER, WF
    KUKOVETZ, WR
    GROSCHNER, K
    BIOCHEMICAL JOURNAL, 1993, 291 : 263 - 267
  • [33] INTRACELLULAR CA2+ INHIBITION OF K+ CHANNELS IN CANINE RENAL-ARTERY - A NOVEL MECHANISM FOR AGONIST-INDUCED MEMBRANE DEPOLARIZED
    GELBAND, CH
    HUME, JR
    CIRCULATION, 1994, 90 (04) : 526 - 526
  • [34] Agonist-induced phosphorylation of the serotonin 5-HT2C receptor regulates its interaction with multiple PDZ protein 1
    Parker, LL
    Backstrom, JR
    Sanders-Bush, E
    Shieh, BH
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2003, 278 (24) : 21576 - 21583
  • [35] THE 2 ISOFORMS OF THE MOUSE SOMATOSTATIN RECEPTOR (MSSTR2A AND MSSTR2B) DIFFER IN COUPLING EFFICIENCY TO ADENYLATE-CYCLASE AND IN AGONIST-INDUCED RECEPTOR DESENSITIZATION
    VANETTI, M
    VOGT, G
    HOLLT, V
    FEBS LETTERS, 1993, 331 (03) : 260 - 266
  • [36] Coupling of c-Src to large conductance voltage- and Ca2+-activated K+ channels as a new mechanism of agonist-induced vasoconstriction
    Alioua, A
    Mahajan, A
    Nishimaru, K
    Zarei, MM
    Stefani, E
    Toro, L
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2002, 99 (22) : 14560 - 14565
  • [37] Differential effect of homozygous haplotypes of the B2-adrenergic receptor (B2AR) and its 5′ promoter on agonist-induced desensititzation in lymphocytes.
    Oostendom, J
    Postma, DS
    Volders, H
    Jongepier, H
    Kauffman, HF
    Nelemans, SA
    Zaagsma, J
    Meurs, H
    NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 2005, 371 (01) : R8 - R8
  • [38] Assessment of striatal D1 and D2 dopamine receptor-G protein coupling by agonist-induced [35S]GTPγS binding
    Geurts, M
    Hermans, E
    Maloteaux, JM
    LIFE SCIENCES, 1999, 65 (16) : 1633 - 1645
  • [39] THE RELATIONSHIP BETWEEN AGONIST-INDUCED ELEVATION OF CYTOSOLIC-FREE CALCIUM ([CA-2+]I) AND MEMBRANE CURRENT IN SINGLE-RAT PAROTID ACINAR-CELLS
    GRAY, PTA
    JOURNAL OF PHYSIOLOGY-LONDON, 1988, 403 : P71 - P71
  • [40] Agonist-induced formation of opioid receptor-G protein-coupled receptor kinase (GRK)-Gβγ complex on membrane is required for GRK2 function in vivo
    Li, JL
    Xiang, B
    Su, WJ
    Zhang, XQ
    Huang, YL
    Ma, L
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2003, 278 (32) : 30219 - 30226