Mathematical analysis of the sodium sensitivity of the human histamine H3 receptor

被引：4
|
作者：
Hans-Joachim Wittmann
Roland Seifert
Andrea Strasser
机构：
[1] University of Regensburg,Faculty of Chemistry and Pharmacy
[2] Medical School of Hannover,Institute of Pharmacology
[3] University of Regensburg,Department of Pharmaceutical and Medicinal Chemistry II, Faculty of Chemistry and Pharmacy
来源：
In Silico Pharmacology | / 2卷 / 1期
关键词：
Histamine H3 receptor; Na+-sensitivity; Mathematical model; Molecular dynamics;
D O I：
10.1186/s40203-014-0001-y
中图分类号：
学科分类号：
摘要：
引用
收藏
相关论文
共 50 条
  • [41] The role of histamine H3 receptor in pancreatic α-cells
    Nakamura, Tadaho
    Yoshikawa, Takeo
    Naganuma, Fumito
    Iida, Tomomitsu
    Miura, Yamato
    Mohsen, Attayeb
    Yanai, Kazuhiko
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2014, 124 : 102P - 102P
  • [42] A scalable synthesis of a histamine H3 receptor antagonist
    Mani, NS
    Jablonowski, JA
    Jones, TK
    JOURNAL OF ORGANIC CHEMISTRY, 2004, 69 (23): : 8115 - 8117
  • [43] Recent progress in histamine H3 receptor chemistry
    Aslanian, R
    Shih, NY
    ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 39, 2004, 39 : 57 - 66
  • [44] Characterization of splicing variants of histamine H3 receptor
    Tanaka, K
    Nakamura, T
    Itadani, H
    Takimura, T
    Hidaka, Y
    Ohta, M
    HISTAMINE RESEARCH IN THE NEW MILLENNIUM, 2001, 1224 : 377 - 382
  • [45] The histamine autoreceptor is a short isoform of the H3 receptor
    Gbahou, F.
    Rouleau, A.
    Arrang, J-M
    BRITISH JOURNAL OF PHARMACOLOGY, 2012, 166 (06) : 1860 - 1871
  • [46] Acidic elements in histamine H3 receptor antagonists
    Sander, Kerstin
    von Coburg, Yvonne
    Camelin, Jean-Claude
    Ligneau, Xavier
    Rau, Oliver
    Schubert-Zsilavecz, Manfred
    Schwartz, Jean-Charles
    Stark, Holger
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (05) : 1581 - 1584
  • [47] Ligand autoradiographical quantification of histamine H3 receptor in human dementia with Lewy bodies
    Lethbridge, Natasha L.
    Chazot, Paul L.
    PHARMACOLOGICAL RESEARCH, 2016, 113 : 245 - 256
  • [48] Structural and Molecular Determinants for Isoform Bias at Human Histamine H3 Receptor Isoforms
    Rahman, Sabrina N.
    McNaught-Flores, Daniel A.
    Huppelschoten, Yara
    Pereira, Daniel da Costa
    Christopoulos, Arthur
    Leurs, Rob
    Langmead, Christopher J.
    ACS CHEMICAL NEUROSCIENCE, 2023, : 645 - 656
  • [49] Molecular cloning and pharmacology of functionally distinct isoforms of the human histamine H3 receptor
    Wellendorph, P
    Goodman, MW
    Burstein, ES
    Nash, NR
    Brann, MR
    Weiner, DM
    NEUROPHARMACOLOGY, 2002, 42 (07) : 929 - 940
  • [50] Histamine H3 receptor-mediated inhibition of noradrenaline release in the human brain
    Schlicker, E
    Werthwein, S
    Zentner, J
    FUNDAMENTAL & CLINICAL PHARMACOLOGY, 1999, 13 (01) : 120 - 122
12345