Recent advances in the synthesis of thiazolo[4,5-b]pyridines. Part 1: Focus on pyridine annulation to thiazole ring (microreview)

被引：1
|
作者：
Chaban, Taras I. [1 ]
Klenina, Olena V. [1 ,3 ]
Chaban, Ihor H. [2 ]
Lelyukh, Maryan I. [2 ]
机构：
[1] Danylo Halytsky Lviv Natl Med Univ, Dept Gen Bioinorgan Phys & Colloidal Chem, 69 Pekarska St, UA-79010 Lvov, Ukraine
[2] Danylo Halytsky Lviv Natl Med Univ, Dept Pharmaceut Organ & Bioorgan Chem, 69 Pekarska St, UA-79010 Lvov, Ukraine
[3] Univ San Pablo CEU, Urbanizac Monteprincipe, Boadilla Del Monte 28668, Spain
来源：
CHEMISTRY OF HETEROCYCLIC COMPOUNDS | 2024年 / 60卷 / 1-2期
关键词：
Compendex;
D O I：
10.1007/s10593-024-03289-0
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The present microreview systematizes recent advances in the synthetic approaches for novel thiazolo[4,5-b]-pyridines and summarizes pharmacological effects they were found to possess. In particular, modern synthetic techniques for thiazolo[4,5-b]pyridine bicyclic scaffold construction starting from thiazole or thiazolidine derivatives followed by pyridine annulation, which results in the target fused thiazolo[4,5-b]pyridines, are analyzed.
引用
收藏
页码：35 / 37
页数：3
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