Reaction of 4-Amino-3-methylthio-5-oxo-6-R-4,5-dihydro-1,2,4-triazines with Sulfonylacetic Acid Nitriles

被引：0
|
作者：
V. N. Britsun
I. M. Bazavova
A. N. Esipenko
M. O. Lozinskii
机构：
[1] Institute of Organic Chemistry,Ukraine National Academy of Sciences
来源：
Chemistry of Heterocyclic Compounds | 2003年 / 39卷 / 12期
关键词：
4-amino-3-methylthio-5-oxo-6-R-4,5-dihydro-1,2,4-triazines; 7-amino-3-R-8-(R'-sulfonyl)-1,4-dihydropyrazolo[5,1-; ][1,2,4]triazin-4-ones; arylsulfonylacetonitriles; dinitriles of sulfonyldiacetic and methylenebis(sulfonylacetic) acids;
D O I：
10.1023/B:COHC.0000018340.15398.18
中图分类号：
学科分类号：
摘要：
The reactions of 4-amino-3-methylthio-5-oxo-6-R-4,5-dihydro-1,2,4-triazines with arylsulfonylacetonitriles and with dinitriles of sulfonyldiacetic acid and methylenebis(sulfonylacetic) acid have been studied. 7-Amino-3-R-8-(R'-sulfonyl)-1,4-dihydropyrazolo[5,1-c][1,2,4]triazin-4-ones have been synthesized and these are the first representatives of geminal sulfones in which the heterocyclic ring is bound directly to the sulfur atoms of the sulfonyl groups.
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页码：1623 / 1626
页数：3
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