Evaluation of some thiophene-based sulfonamides as potent inhibitors of carbonic anhydrase I and II isoenzymes isolated from human erythrocytes by kinetic and molecular modelling studies

被引：0

作者：

Zuhal Alım

Zeynep Köksal

Muhammet Karaman

机构：

[1] Kırşehir Ahi Evran University,Department of Chemistry, Faculty of Science and Arts

[2] Istanbul Medeniyet University,Department of Chemistry, Faculty of Engineering and Natural Sciences

[3] Kilis 7 Aralık University,Department of Molecular Biology and Genetics, Faculty of Arts and Sciences

来源：

Pharmacological Reports | 2020年 / 72卷

关键词：

Thiophene; Sulfonamide; Carbonic anhydrase; Inhibition; Molecular modelling;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

引用

页码：1738 / 1748

页数：10

共 21 条

[1] Evaluation of some thiophene-based sulfonamides as potent inhibitors of carbonic anhydrase I and II isoenzymes isolated from human erythrocytes by kinetic and molecular modelling studies
Alim, Zuhal
Koksal, Zeynep
Karaman, Muhammet
PHARMACOLOGICAL REPORTS, 2020, 72 (06) : 1738 - 1748
[2] Inhibition properties of some flavonoids on carbonic anhydrase I and II isoenzymes purified from human erythrocytes
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Beydemir, Sukru
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JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY, 2017, 31 (09)
[3] Sulfonamides incorporating piperazine bioisosteres as potent human carbonic anhydrase I, II, IV and IX inhibitors
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Picchioni, Ilaria
Bartolucci, Gianluca
Braconi, Laura
Dei, Silvia
Teodori, Elisabetta
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Romanelli, Maria Novella
BIOORGANIC CHEMISTRY, 2019, 91
[4] Kinetic and in silico studies of hydroxy-based inhibitors of carbonic anhydrase isoforms I and II
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[5] Inhibition Profiles of Some Symmetric Sulfamides Derived from Phenethylamines on Human Carbonic Anhydrase I, and II Isoenzymes
Topal, Fevzi
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Tumer, Ferhan
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CHEMISTRY & BIODIVERSITY, 2021, 18 (10)
[6] Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity
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Carta, Fabrizio
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JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY, 2025, 39 (01)
[7] Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and molecular docking studies
Eldehna, Wagdy M.
Al-Ansary, Ghada H.
Bua, Silvia
Nocentini, Alessio
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 127 : 521 - 530
[8] Nimesulide linked acyl thioureas potent carbonic anhydrase I, II and α-glucosidase inhibitors: Design, synthesis and molecular docking studies
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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS, 2022, 6
[9] Synthesis, characterization and biological evaluation of pyrazole-based benzene sulfonamides as inhibitors of human carbonic anhydrase II, IX and XII
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Ullah, Saif
Alrokayan, Salman
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RSC ADVANCES, 2023, 13 (27) : 18461 - 18479
[10] Chalcone-based benzenesulfonamides as potent and selective inhibitors for human carbonic anhydrase II: Design, synthesis, in vitro, and in silico studies
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