Hit-to-lead optimization of amino-carboxamide benzothiazoles as LSD1 inhibitors

被引:0
|
作者
Du’a Al bustanji
Soraya Alnabulsi
Enas A. Al-Hurani
机构
[1] Jordan University of Science and Technology,Department of Medicinal Chemistry and Pharmacognosy, Faculty of Pharmacy
[2] P.O. Box 3030,undefined
来源
Medicinal Chemistry Research | 2023年 / 32卷
关键词
LSD1 enzyme; hit-to-lead optimization; anticancer; structure-activity relationship; amino-carboxamide benzothiazoles.;
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页码:910 / 929
页数:19
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