Design, synthesis, and preliminary pharmacological evaluation of novel thiazolidinone derivatives as potential benzodiazepine agonists

被引:0
|
作者
Ali Almasirad
Maryam Ghadimi
Saeideh Mirahmadi
Pouya Ahmadian Kodakan
Reza Jahani
Maryam Nazari
Elham Rezaee
Homa Azizian
Parmida Rabizadeh
Sayyed Abbas Tabatabai
Mehrdad Faizi
机构
[1] Islamic Azad University,Department of Medicinal Chemistry, Faculty of Pharmacy, Tehran Medical Sciences
[2] Shahid Beheshti University of Medical Sciences,Department of Pharmacology and Toxicology, School of Pharmacy
[3] Shahid Beheshti University of Medical Sciences,Department of Pharmaceutical Chemistry, School of Pharmacy
[4] Iran University of Medical Sciences,Department of Medicinal Chemistry, Pharmacy School, International Vice Chancellor Office
来源
Molecular Diversity | 2022年 / 26卷
关键词
Anticonvulsant; Benzodiazepine; 4-Thiazolidinone derivatives; Synthesis;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:769 / 780
页数:11
相关论文
共 50 条
  • [41] Design and synthesis of novel 1,4-benzodiazepine derivatives and their biological evaluation as cholinesterase inhibitors
    Mohamed, Lamia W.
    El-yamany, Mohamed F.
    ARCHIVES OF PHARMACAL RESEARCH, 2012, 35 (08) : 1369 - 1377
  • [42] Design and synthesis of novel 1,4-benzodiazepine derivatives and their biological evaluation as cholinesterase inhibitors
    Lamia Wagdy Mohamed
    Mohamed F. El-yamany
    Archives of Pharmacal Research, 2012, 35 : 1369 - 1377
  • [43] Design, synthesis and preliminary pharmacological evaluation of new piperidine and piperazine derivatives as cognition-enhancers
    Martini, Elisabetta
    Ghelardini, Carla
    Dei, Silvia
    Guandalini, Luca
    Manetti, Dina
    Melchiorre, Michele
    Norcini, Monica
    Scapecchi, Serena
    Teodori, Elisabetta
    Romanelli, Maria Novella
    BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (03) : 1431 - 1443
  • [44] Synthesis and Pharmacological Evaluation of Novel Quinazoline Derivatives as Potential EGFR Inhibitors for Breast Cancer
    Dwivedi, Deepak K.
    Agrawal, Ram Kishore
    INTERNATIONAL JOURNAL OF PHARMACEUTICAL INVESTIGATION, 2023, 13 (01) : 82 - 86
  • [45] Design, synthesis, molecular docking and pharmacological evaluation of novel triazine-based triazole derivatives as potential anticonvulsant agents
    Alhamzani, Abdulrahman G.
    Yousef, Tarek A.
    Abou-Krisha, Mortaga M.
    Raghu, M. S.
    Kumar, K. Yogesh
    Prashanth, M. K.
    Jeon, Byong-Hun
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2022, 77
  • [46] Design, Synthesis, and Pharmacological Screening of Novel Porphyrin Derivatives
    Fadda, Ahmed A.
    El-Mekawy, Rasha E.
    El-Shafei, Ahmed
    Freeman, Harold S.
    Hinks, David
    El-Fedawy, Andmanal
    JOURNAL OF CHEMISTRY, 2013, 2013
  • [47] Mixed κ agonists and μ agonists/antagonists as potential pharmacotherapeutics for cocaine abuse:: Synthesis and pharmacological evaluation of N-substituted derivatives of morphinan.
    Gu, XH
    Bidlack, JM
    van Vliet, LA
    Negas, SS
    Mello, NK
    Neumeyer, JL
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 222 : U676 - U676
  • [48] Design, Synthesis, and Evaluation of Novel Strobilurins Derivatives as Potential Fungicidal Agents
    Wang, Xianyou
    Liu, Xin
    Zheng, Jiayan
    Pang, Yanping
    Zhao, Xin
    Wu, Guangchen
    Zhao, Zhilei
    INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY, 2021, 31 (04) : 613 - 619
  • [49] Design, synthesis and preliminary evaluation of novel pyrrolidine derivatives as matrix metalloproteinase inhibitors
    Cheng, Xian-Chao
    Wang, Qiang
    Fang, Hao
    Tang, Wei
    Xu, Wen-Fang
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2008, 43 (10) : 2130 - 2139
  • [50] Design, synthesis, and preliminary biological evaluation of novel ketone derivatives of shikimic acid
    Jiang, Min
    Xiong, Bing
    Shen, Yu-mei
    Yang, Chunhao
    RSC ADVANCES, 2013, 3 (43): : 20599 - 20605