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- [21] A phase I dose escalation study of oral MK-2206 (allosteric Akt inhibitor) with oral selumetinib (AZD6244; ARRY-142866) (MEK 1/2 inhibitor) in patients with advanced or metastatic solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2012, 30 (15)Khan, Khurum Hayat论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAYan, Li论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAMezynski, Janusz论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAMoreno, Victor论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAGarrett, Chris R.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAOng, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAShannon, Keith A.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USAMorosky, Anne论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USARubin, Eric H.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USATetteh, Ernestina论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USASkolnik, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USASmith, Ian C.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USASmith, Paul D.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USADe Bono, Johann Sebastian论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USATolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: Merck Sharp & Dohme Ltd, N Wales, PA USA
- [22] Interrogating Two Schedules of the AKT Inhibitor MK-2206 in Patients with Advanced Solid Tumors Incorporating Novel Pharmacodynamic and Functional Imaging BiomarkersCLINICAL CANCER RESEARCH, 2014, 20 (22) : 5672 - 5685Yap, Timothy A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, England Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandYan, Li论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Whitehouse Stn, NJ USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandPatnaik, Amita论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, San Antonio, TX USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandTunariu, Nina论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Radiotherapy & Imaging, CR UK & EPSRC Canc Imaging Ctr, Sutton, Surrey, England Royal Marsden NHS Fdn Trust, Sutton SM2 5PT, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandBiondo, Andrea论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, England Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandFearen, Ivy论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Whitehouse Stn, NJ USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandPapadopoulos, Kyriakos P.论文数: 0 引用数: 0 h-index: 0机构: South Texas Accelerated Res Therapeut, San Antonio, TX USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandOlmos, David论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, England Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandBaird, Richard论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, England Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandDelgado, Liliana论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Whitehouse Stn, NJ USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandTetteh, Ernestina论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Whitehouse Stn, NJ USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandBeckman, Robert A.论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Whitehouse Stn, NJ USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandLupinacci, Lisa论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Whitehouse Stn, NJ USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandRiisnaes, Ruth论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandDecordova, Shaun论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandHeaton, Simon P.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandSwales, Karen论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglanddeSouza, Nandita M.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Radiotherapy & Imaging, CR UK & EPSRC Canc Imaging Ctr, Sutton, Surrey, England Royal Marsden NHS Fdn Trust, Sutton SM2 5PT, Surrey, England H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandLeach, Martin O.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Radiotherapy & Imaging, CR UK & EPSRC Canc Imaging Ctr, Sutton, Surrey, England Royal Marsden NHS Fdn Trust, Sutton SM2 5PT, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandGarrett, Michelle D.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandSullivan, Daniel M.论文数: 0 引用数: 0 h-index: 0机构: H Lee Moffitt Canc Ctr & Res Inst, Tampa, FL USA Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, Englandde Bono, Johann S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, England Inst Canc Res, Div Clin Studies, Surrey, England Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, EnglandTolcher, Anthony W.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden NHS Fdn Trust, Drug Dev Unit, Sutton SM2 5PT, Surrey, England
- [23] Phase I clinical trial of an allosteric AKT inhibitor, MK-2206, using a once weekly (QW) dose regimen in patients with advanced solid tumors.JOURNAL OF CLINICAL ONCOLOGY, 2011, 29 (15)Biondo, A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandYap, T. A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandYan, L.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandPatnaik, A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandFearen, I.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandBaird, R. D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandPapadopoulos, K. P.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandDelgado, L. M.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandTaylor, A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandLupinacci, L.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandBlackman, S. C.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandDecordova, S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandTall, M.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandHeaton, S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandGarrett, M. D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandSullivan, D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandDe Bono, J. S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, EnglandTolcher, A. W.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp, Sutton, Surrey, England
- [24] Phase I Study of an AKT Inhibitor (MK-2206) Combined with Lapatinib in Adult Solid Tumors Followed by Dose Expansion in Advanced HER2+ Breast CancerCLINICAL CANCER RESEARCH, 2016, 22 (11) : 2659 - 2667Wisinski, Kari B.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USATevaarwerk, Amye J.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USABurkard, Mark E.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USARampurwala, Murtuza论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USAEickhoff, Jens论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Dept Biostat & Med Informat, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USABell, Maria C.论文数: 0 引用数: 0 h-index: 0机构: Sanford Canc Ctr, Sioux Falls, SD USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USAKolesar, Jill M.论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Pharm, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USAFlynn, Christopher论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USALiu, Glenn论文数: 0 引用数: 0 h-index: 0机构: Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA Univ Wisconsin, Sch Med & Publ Hlth, Madison, WI 53705 USA Univ Wisconsin, Carbone Canc Ctr, 1111 Highland Ave, Madison, WI 53705 USA
- [25] Phase II study of the oral AKT inhibitor, MK-2206, for acute myeloid leukemia (AML) in second relapse.CANCER RESEARCH, 2013, 73 (08)Konopleva, Marina Y.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAWalter, Roland B.论文数: 0 引用数: 0 h-index: 0机构: Fred Hutchinson Canc Res Ctr, Seattle, WA 98104 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAFaderl, Stefan论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAJabbour, Elias论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAZeng, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABorthakur, Gautam论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USARuvolo, Peter论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAHuang, Xuelin论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKadia, Tapan论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAFeliu, Jennie论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABurger, Jan A.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAAndreeff, Michael论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USALiu, Wenbin论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKornblau, Steven M.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USABaggerly, Keith论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAEstey, Elihu论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Sch Med, Seattle, WA USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USAKantarjian, Hagop论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Houston, TX 77030 USA
- [26] Discovery of MK-2206: The first oral allosteric Akt kinase inhibitor for the treatment of cancerABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 244Kelly, Michael J., III论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA Merck & Co Inc, Dept Med Chem, West Point, PA 19486 USA
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