Catalyst-free tandem Michael addition-cyclization reactions in aqueous media for the synthesis of benzimidazo[1,2-a]pyrimidinone derivatives

被引：0

作者：

ChuanLi Ren

Yan Wang

Dong Wang

YongJun Chen

Li Liu

机构：

[1] Chinese Academy of Sciences,Beijing National Laboratory (BNLMS), CAS Key Laboratory for Molecular Recognition and Function

[2] Chinese Academy of Sciences,Institute of Chemistry

来源：

Science China Chemistry | 2010年 / 53卷

关键词：

queous media; Baylis-Hillman alcohol; 2-aminobenzimidazole; pesticidal activity;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

The catalyst-free reactions of Baylis-Hillman alcohols (1a-i) with 2-aminobenzimidazole (2) in THF-H2O (1:4) were developed for the convenient and greener synthesis of benzimidazo[1,2-a]pyrimidinone derivatives (3a-i). The pesticidal activities of 3a-i were examined to investigate a new biological activity of the imidazo[1,2-a]pyrimidinone-type compounds.

引用

页码：1492 / 1496

页数：4

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