Cariprazine (RGH-188), a D3-preferring dopamine D3/D2 receptor partial agonist antipsychotic candidate demonstrates anti-abuse potential in rats

被引:0
|
作者
V. Román
I. Gyertyán
K. Sághy
B. Kiss
Zs. Szombathelyi
机构
[1] Gedeon Richter Plc,Pharmacology and Drug Safety Research
[2] Gedeon Richter Plc.,Department of Behavioural Pharmacology
来源
Psychopharmacology | 2013年 / 226卷
关键词
Cariprazine; Aripiprazole; Bifeprunox; Dopamine receptor; Cocaine self-administration; Cocaine seeking; Relapse; Antipsychotic; Antimanic;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:285 / 293
页数:8
相关论文
共 50 条
  • [1] Cariprazine (RGH-188), a D3-preferring dopamine D3/D2 receptor partial agonist antipsychotic candidate demonstrates anti-abuse potential in rats
    Roman, V.
    Gyertyan, I.
    Saghy, K.
    Kiss, B.
    Szombathelyi, Zs.
    PSYCHOPHARMACOLOGY, 2013, 226 (02) : 285 - 293
  • [2] CARIPRAZINE, A D3-PREFERRING DOPAMINE D3/D2 RECEPTOR PARTIAL AGONIST ANTIPSYCHOTIC CANDIDATE DEMONSTRATES ANTI-ABUSE POTENTIAL IN RATS
    Gyertyan, Istvan
    Roman, V.
    Saghy, K.
    Kiss, B.
    Szombathelyi, Z.
    SCHIZOPHRENIA BULLETIN, 2011, 37 : 288 - 289
  • [3] Cariprazine (RGH-188), a Dopamine D3 Receptor-Preferring, D3/D2 Dopamine Receptor Antagonist-Partial Agonist Antipsychotic Candidate: In Vitro and Neurochemical Profile
    Kiss, Bela
    Horvath, Attila
    Nemethy, Zsolt
    Schmidt, Eva
    Laszlovszky, Istvan
    Bugovics, Gyula
    Fazekas, Karoly
    Hornok, Katalin
    Orosz, Szabolcs
    Gyertyan, Istvan
    Agai-Csongor, Eva
    Domany, Gyoergy
    Tihanyi, Karoly
    Adham, Nika
    Szombathelyi, Zsolt
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2010, 333 (01): : 328 - 340
  • [4] RGH-188, a d3/d2 dopamine receptor antagonist/partial agonist atypical antipsychotic candidate
    Laszlovszky, I.
    Kiss, B.
    Gyertyan, I.
    Meszaros, G. Pasztor
    Seneca, N.
    Schmidt, E.
    Nemethy, Z. S.
    Bugovics, G. Y.
    Saghy, K.
    Laszy, J.
    Kapas, M.
    Nemeth, G. Y.
    Szombathelyi, Z. S.
    EUROPEAN PSYCHIATRY, 2008, 23 : S163 - S163
  • [5] Favourable behavioural actions of RGH-188, a novel dopamine D3/D2 receptor antagonist/partial agonist antipsychotic candidate
    Gyertyan, I.
    Kiss, B.
    Saghy, K.
    Laszy, J.
    Szabo, G.
    Agai-Csongor, E.
    Domany, G.
    Tihanyi, K.
    Szombathelyi, Z.
    BEHAVIOURAL PHARMACOLOGY, 2007, 18 : S12 - S13
  • [6] Discovery of cariprazine (RGH-188): A novel antipsychotic acting on dopamine D3/D2 receptors
    Agai-Csongor, Eva
    Domany, Gyoergy
    Nogradi, Katalin
    Galambos, Janos
    Vago, Istvan
    Keseru, Gyoergy Miklos
    Greiner, Istvan
    Laszlovszky, Istvan
    Gere, Aniko
    Schmidt, Eva
    Kiss, Bela
    Vastag, Monika
    Tihanyi, Karoly
    Saghy, Katalin
    Laszy, Judit
    Gyertyan, Istvan
    Zajer-Balazs, Maria
    Gemesi, Larisza
    Kapas, Margit
    Szombathelyi, Zsolt
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (10) : 3437 - 3440
  • [7] RGH-188, a D3/D2 dopamine receptor partial agonist antipsychotic candidate with excellent brain availability and low EPS liability
    Gyertyan, Istvan
    Kiss, Bela
    Saghy, Katalin
    Pasztor, Gabriella
    Gemesi, Larisza I.
    Kapas, Margit
    Agai-Csongor, Eva
    Domany, Gyorgy
    Tihanyi, Karoly
    Szombathelyi, Zsolt
    BIOLOGICAL PSYCHIATRY, 2007, 61 (08) : 76S - 76S
  • [8] Pharmacokinetics of RGH-188, a novel dopamine D3/D2 antagonist/partial agonist atypical antipsychotic, in rats and dogs
    Meszaros, G. Pasztor
    Bolf, E. Terjeki
    Gemesi, L.
    Kapas, M.
    Tihanyi, K.
    Szombathelyi, Z.
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2008, 18 : S456 - S457
  • [9] Pharmacological profile of RGH-188, a novel dopamine D3/D2 receptor antagonist/partial agonist atypical antipsychotic
    Gyertyan, I.
    Kiss, B.
    Saghy, K.
    Laszlovszky, I.
    Horvath, A.
    Laszy, J.
    Schmidt, E.
    Szabo, G.
    Domany, G.
    Csongor, E. Agai
    Tihanyi, K.
    Szombathelyi, Z.
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2006, 16 : S432 - S432
  • [10] Dopamine 1321133 receptor occupancy of RGH-188, a D3/D2 antagonist/partial agonist antipsychotic, in healthy volunteers
    Laszovszky, I.
    Nemeth, G.
    Meszaros, G. Pasztor
    Kapas, M.
    Brooks, D. J.
    Pavese, N.
    Szombathelyi, Z.
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2007, 17 : S455 - S455