Synthesis of 2,5-di(hydroxyalkyl)-1,3-thiazoles

被引：0
|
作者：
V. O. Sinenko
S. R. Slivchuk
Ya. G. Bal’on
V. S. Brovarets
机构：
[1] National Academy of Sciences of Ukraine,Institute of Bioorganic Chemistry and Petrochemistry
[2] National Academy of Medical Science,Komisarenko Institute of Endocrinology and Metabolism
来源：
Russian Journal of General Chemistry | 2015年 / 85卷
关键词：
1,3-thiazole; -butyllithium; electrophile; diol;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
A general approach towards synthesis of 2(5)-hydroxyalkyl-substituted 1,3-thiazole derivatives has been proposed. The method includes lithiation of 1,3-thiazole ring followed by reacting the formed thiazole lithium derivatives with electrophiles.
引用
收藏
页码：1855 / 1861
页数：6
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