Synthesis and antituberculosis activity of certain steroidal derivatives of the 5α-series

被引:0
|
作者
M. I. Merlani
L. Sh. Amiranashvili
K. G. Mulkidzhanyan
A. R. Shelar
F. V. Manvi
机构
[1] Academy of Sciences of Georgia,I. G. Kutateladze Institute of Pharmaceutical Chemistry
[2] University KLES,Pharmaceutical College
来源
关键词
antituberculosis activity; isonicotinoylhydrazones; thiosemicarbazones; steroids;
D O I
暂无
中图分类号
学科分类号
摘要
The antituberculosis activity of several steroidal compounds of various structure was studied. Severa compounds that were active toward M. tuberculosis were found in in vitro tests.
引用
收藏
页码:618 / 620
页数:2
相关论文
共 50 条
  • [31] Design, synthesis and cytotoxic activity of a novel series of steroidal phenylpyrazoles
    Li, Jian
    Zhao, Ximei
    Li, Longbo
    Yuan, Zhipeng
    Tan, Fangfang
    Shi, Baojun
    Zhang, Jiwen
    STEROIDS, 2016, 107 : 45 - 54
  • [32] Synthesis and Structure Activity Relationship of Organometallic Steroidal Androgen Derivatives
    Top, Siden
    Thibaudeau, Celine
    Vessieres, Anne
    Brule, Emilie
    Le Bideau, Franck
    Joerger, Jean-Michel
    Plamont, Marie-Aude
    Samreth, Soth
    Edgar, Alan
    Marrot, Jerome
    Herson, Patrick
    Jaouen, Gerard
    ORGANOMETALLICS, 2009, 28 (05) : 1414 - 1424
  • [33] Synthesis and in vitro antimicrobial activity of new steroidal hydrazone derivatives
    Mistry, Shailesh
    Singh, Akhilesh Kumar
    FUTURE JOURNAL OF PHARMACEUTICAL SCIENCES, 2022, 8 (01)
  • [34] Synthesis and antitumor activity of novel steroidal imidazolium salt derivatives
    Deng, Guogang
    Zhou, Bei
    Wang, Jing
    Chen, Zhuo
    Gong, Liang
    Gong, Yaxiao
    Wu, Dongmei
    Li, Yan
    Zhang, Hongbin
    Yang, Xiaodong
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2019, 168 : 232 - 252
  • [35] Synthesis and in vitro antibacterial activity of new steroidal thiosemicarbazone derivatives
    Khan, Salman Ahmad
    Kumar, Praveen
    Joshi, Rajkumar
    Iqbal, Prince F.
    Saleem, Kishwar
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2008, 43 (09) : 2029 - 2034
  • [36] Synthesis and in vitro antimicrobial activity of new steroidal hydrazone derivatives
    Shailesh Mistry
    Akhilesh Kumar Singh
    Future Journal of Pharmaceutical Sciences, 8
  • [37] Synthesis, Toxicity, and Antituberculosis Activity of Isoniazid Derivatives Containing Sterically Hindered Phenols
    Yu. N. Oludina
    A. D. Voloshina
    M. V. Kulik
    V. V. Zobov
    S. V. Bukharov
    R. G. Tagasheva
    G. N. Nugumanova
    A. R. Burilov
    M. A. Kravchenko
    S. N. Skornyakov
    G. L. Rusinov
    Pharmaceutical Chemistry Journal, 2014, 48 : 5 - 7
  • [38] Synthesis and antibacterial activity of a series novel 5,7-diisoprenyloxyflavone derivatives
    Jin, Qing-Hao
    Fu, Zhi-Yang
    Xia, Ya-Nan
    Liu, Bing-Yu
    Jiang, Hai-Ying
    BRAZILIAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2020, 56
  • [39] SYNTHESIS AND ANTITUBERCULOSIS ACTIVITY OF DERIVATIVES OF THE DITERPENOID ISOSTEVIOL WITH AZINE, HYDRAZIDE, AND HYDRAZONE MOIETIES
    Garifullin, B. F.
    Strobykina, I. Yu
    Mordovskoi, G. G.
    Mironov, V. F.
    Kataev, V. E.
    CHEMISTRY OF NATURAL COMPOUNDS, 2011, 47 (01) : 55 - 58
  • [40] Synthesis, Toxicity, and Antituberculosis Activity of Isoniazid Derivatives Containing Sterically Hindered Phenols
    Oludina, Yu. N.
    Voloshina, A. D.
    Kulik, M. V.
    Zobov, V. V.
    Bukharov, S. V.
    Tagasheva, R. G.
    Nugumanova, G. N.
    Burilov, A. R.
    Kravchenko, M. A.
    Skornyakov, S. N.
    Rusinov, G. L.
    PHARMACEUTICAL CHEMISTRY JOURNAL, 2014, 48 (01) : 5 - 7