N-Propargyltetrahydrocarbazoles and N-propargyltetrahydro-γ-carbolines in 1,3-cycloaddition with azide-containing pharmacophores

被引：0

作者：

V. B. Sokolov

A. Yu. Aksinenko

T. A. Epishina

T. V. Goreva

机构：

[1] Russian Academy of Sciences,Institute of Physiologically Active Compounds

来源：

Russian Chemical Bulletin | 2019年 / 68卷

关键词：

carbazoles; tetrahydrocarbazoles; tetrahydro-γ-carbolines; 1-aminoadamantanes; phenothiazines; copper-catalyzed 1,3-dipolar cycloaddition; 1,2,3-triazoles; alkynes; azides;

D O I：

暂无

中图分类号：

学科分类号：

摘要：

A modification of tetrahydrocarbazoles and tetrahydro-γ-carbolines with pharmacophore ligands was performed based on the copper-catalyzed 1,3-dipolar cycloaddition of their N-propargyl derivatives to azide-containing carbazoles, tetrahydrocarbazoles, 1-aminoadamantanes, and phenothiazine.

引用

页码：1424 / 1428

页数：4

共 29 条

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