N-Propargyltetrahydrocarbazoles and N-propargyltetrahydro-γ-carbolines in 1,3-cycloaddition with azide-containing pharmacophores

被引：0
|
作者：
V. B. Sokolov
A. Yu. Aksinenko
T. A. Epishina
T. V. Goreva
机构：
[1] Russian Academy of Sciences,Institute of Physiologically Active Compounds
来源：
Russian Chemical Bulletin | 2019年 / 68卷
关键词：
carbazoles; tetrahydrocarbazoles; tetrahydro-γ-carbolines; 1-aminoadamantanes; phenothiazines; copper-catalyzed 1,3-dipolar cycloaddition; 1,2,3-triazoles; alkynes; azides;
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学科分类号：
摘要：
A modification of tetrahydrocarbazoles and tetrahydro-γ-carbolines with pharmacophore ligands was performed based on the copper-catalyzed 1,3-dipolar cycloaddition of their N-propargyl derivatives to azide-containing carbazoles, tetrahydrocarbazoles, 1-aminoadamantanes, and phenothiazine.
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页码：1424 / 1428
页数：4
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