The synthesis and investigation of the antimicrobial activity of some new phenylselanyl-1-(toluene-4-sulfonyl)-1H-tetrazole derivatives

被引：0
|
作者：
Yılmaz Yıldırır
M. Faruk Us
Naki Çolak
Hamdi Özkan
Serkan Yavuz
Ali Disli
Sahlan Ozturk
Lemi Turker
机构：
[1] Gazi University,Faculty of Science and Arts, Chemistry Department
[2] Central Veterinary Controls and Research Institute,Faculty of Science and Arts, Biology Department
[3] Gazi University,Faculty of Science and Arts, Chemistry Department
[4] Middle East Technical University,undefined
来源：
Medicinal Chemistry Research | 2009年 / 18卷
关键词：
Tetrazole toluenesulfonic acid; Antimicrobial activity; SMX; SRZ;
D O I：
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中图分类号：
学科分类号：
摘要：
The sulfonamide functional group has aroused interest in both medicinal and bioorganic chemistry. In this study, some new phenylselanyl–1–(toluene-4-sulfonyl)-1H-tetrazole derivatives (2a–f) have been synthesized using dicyclohexylcarbodiimide/dimethylaminopyridine (DCC/DMAP). The structures of the presently synthesized compounds were elucidated by spectroscopic methods [Fourier-transform infrared (FTIR) spectroscopy, 1H nuclear magnetic resonance (NMR), 13C nuclear magnetic resonance-attached proton test (13C NMR-APT), and mass spectrometry (MS)]. In addition, the antimicrobial activity of the synthesized compounds and two antibiotics [sulfamethoxazole (SMX) and sulfamerazine (SRZ)] were investigated against some microorganisms.
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页码：91 / 97
页数：6
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