共 50 条
- [41] Substituted bisaryl benzamide derivatives to inhibit HIV-1 replicationABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 251Malik, Neha论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Evanston, IL USA Northwestern Univ, Evanston, IL USASchiltz, Gary论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Evanston, IL USA Northwestern Univ, Evanston, IL USASong, Chisu论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Evanston, IL USA Northwestern Univ, Evanston, IL USAD'Aquila, Richard论文数: 0 引用数: 0 h-index: 0机构: Northwestern Univ, Evanston, IL USA Northwestern Univ, Evanston, IL USA
- [42] Styrylquinoline derivatives:: A new class of potent HIV-1 integrase inhibitors that block HIV-1 replication in CEM cellsJOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (15) : 2846 - 2857Mekouar, K论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, FranceMouscadet, JF论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, FranceDesmaële, D论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, FranceSubra, F论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, FranceLeh, H论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, FranceSavouré, D论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, FranceAuclair, C论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, Franced'Angelo, J论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Sud, Ctr Etud Pharmaceut, URA CNRS 1843, Unite Chim Organ, F-92296 Chatenay Malabry, France
- [43] A Symmetric Region of the HIV-1 Integrase Dimerization Interface Is Essential for Viral ReplicationPLOS ONE, 2012, 7 (09):Serrao, Erik论文数: 0 引用数: 0 h-index: 0机构: Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USA Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USAThys, Wannes论文数: 0 引用数: 0 h-index: 0机构: Katholieke Univ Leuven, Lab Mol Virol & Gene Therapy, Div Mol Med, Flanders, Belgium Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USADemeulemeester, Jonas论文数: 0 引用数: 0 h-index: 0机构: Katholieke Univ Leuven, Lab Mol Virol & Gene Therapy, Div Mol Med, Flanders, Belgium Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USAAl-Mawsawi, Laith Q.论文数: 0 引用数: 0 h-index: 0机构: Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USA Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USAChrist, Frauke论文数: 0 引用数: 0 h-index: 0机构: Katholieke Univ Leuven, Lab Mol Virol & Gene Therapy, Div Mol Med, Flanders, Belgium Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USADebyser, Zeger论文数: 0 引用数: 0 h-index: 0机构: Katholieke Univ Leuven, Lab Mol Virol & Gene Therapy, Div Mol Med, Flanders, Belgium Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USANeamati, Nouri论文数: 0 引用数: 0 h-index: 0机构: Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USA Univ So Calif, Sch Pharm, Dept Pharmacol & Pharmaceut Sci, Los Angeles, CA 90089 USA
- [44] Uncommon Pathways of Immune Escape Attenuate HIV-1 Integrase Replication CapacityJOURNAL OF VIROLOGY, 2012, 86 (12) : 6913 - 6923Brockman, Mark A.论文数: 0 引用数: 0 h-index: 0机构: Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada British Columbia Ctr Excellence HIV AIDS, Vancouver, BC, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaChopera, Denis R.论文数: 0 引用数: 0 h-index: 0机构: Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaOlvera, Alex论文数: 0 引用数: 0 h-index: 0机构: AIDS Res Inst IrsiCaixa, Badalona, Spain Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaBrumme, Chanson J.论文数: 0 引用数: 0 h-index: 0机构: British Columbia Ctr Excellence HIV AIDS, Vancouver, BC, Canada Univ British Columbia, Vancouver, BC V5Z 1M9, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaSela, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Ragon Inst MGH MIT & Harvard, Boston, MA USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaMarkle, Tristan J.论文数: 0 引用数: 0 h-index: 0机构: Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaMartin, Eric论文数: 0 引用数: 0 h-index: 0机构: Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaCarlson, Jonathan M.论文数: 0 引用数: 0 h-index: 0机构: Microsoft Res, Los Angeles, CA USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaLe, Anh Q.论文数: 0 引用数: 0 h-index: 0机构: Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaMcGovern, Rachel论文数: 0 引用数: 0 h-index: 0机构: British Columbia Ctr Excellence HIV AIDS, Vancouver, BC, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaCheung, Peter K.论文数: 0 引用数: 0 h-index: 0机构: British Columbia Ctr Excellence HIV AIDS, Vancouver, BC, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaKelleher, Anthony D.论文数: 0 引用数: 0 h-index: 0机构: Univ New S Wales, Kirby Inst, Sydney, NSW, Australia Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaJessen, Heiko论文数: 0 引用数: 0 h-index: 0机构: Jessen Praxis, Berlin, Germany Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaMarkowitz, Martin论文数: 0 引用数: 0 h-index: 0机构: Aaron Diamond AIDS Res Ctr, New York, NY USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaRosenberg, Eric论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Boston, MA 02114 USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaFrahm, Nicole论文数: 0 引用数: 0 h-index: 0机构: Fred Hutchinson Canc Res Ctr, Seattle, WA 98104 USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaSanchez, Jorge论文数: 0 引用数: 0 h-index: 0机构: Asociac Civil IMPACTA Salud & Educ, Lima, Peru Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada论文数: 引用数: h-index:机构:John, Mina论文数: 0 引用数: 0 h-index: 0机构: Murdoch Univ, Perth, WA, Australia Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaHarrigan, P. Richard论文数: 0 引用数: 0 h-index: 0机构: British Columbia Ctr Excellence HIV AIDS, Vancouver, BC, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaHeckerman, David论文数: 0 引用数: 0 h-index: 0机构: Microsoft Res, Los Angeles, CA USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaBrander, Christian论文数: 0 引用数: 0 h-index: 0机构: AIDS Res Inst IrsiCaixa, Badalona, Spain ICREA, Barcelona, Spain Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaWalker, Bruce D.论文数: 0 引用数: 0 h-index: 0机构: Ragon Inst MGH MIT & Harvard, Boston, MA USA Simon Fraser Univ, Burnaby, BC V5A 1S6, CanadaBrumme, Zabrina L.论文数: 0 引用数: 0 h-index: 0机构: Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada British Columbia Ctr Excellence HIV AIDS, Vancouver, BC, Canada Simon Fraser Univ, Burnaby, BC V5A 1S6, Canada
- [45] Dual inhibition of HIV-1 replication by integrase-LEDGF allosteric inhibitors is predominant at the post-integration stageRetrovirology, 10Erwann Le Rouzic论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSDamien Bonnard论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSSophie Chasset论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSJean-Michel Bruneau论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSFrancis Chevreuil论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSFrédéric Le Strat论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSJuliette Nguyen论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSRoxane Beauvoir论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSCéline Amadori论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSJulie Brias论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSSophie Vomscheid论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSSylvia Eiler论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSNicolas Lévy论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSOlivier Delelis论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSEric Deprez论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSAli Saïb论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSAlessia Zamborlini论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSStéphane Emiliani论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSMarc Ruff论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSBenoit Ledoussal论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSFrançois Moreau论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRSRichard Benarous论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis,IGBMC, Inserm, CNRS
- [46] Dual inhibition of HIV-1 replication by integrase-LEDGF allosteric inhibitors is predominant at the post-integration stageRETROVIROLOGY, 2013, 10Le Rouzic, Erwann论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceBonnard, Damien论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceChasset, Sophie论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceBruneau, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceChevreuil, Francis论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceLe Strat, Frederic论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceNguyen, Juliette论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceBeauvoir, Roxane论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceAmadori, Celine论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceBrias, Julie论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceVomscheid, Sophie论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceEiler, Sylvia论文数: 0 引用数: 0 h-index: 0机构: Univ Strasbourg, CNRS, INSERM, IGBMC, F-67404 Illkirch Graffenstaden, France Biodim Mutabilis, F-93230 Romainville, FranceLevy, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Univ Strasbourg, CNRS, INSERM, IGBMC, F-67404 Illkirch Graffenstaden, France Biodim Mutabilis, F-93230 Romainville, FranceDelelis, Olivier论文数: 0 引用数: 0 h-index: 0机构: CNRS, ENS Cachan, LBPA, Cachan, France Biodim Mutabilis, F-93230 Romainville, FranceDeprez, Eric论文数: 0 引用数: 0 h-index: 0机构: CNRS, ENS Cachan, LBPA, Cachan, France Biodim Mutabilis, F-93230 Romainville, FranceSaib, Ali论文数: 0 引用数: 0 h-index: 0机构: Univ Paris Diderot, Conservatoire Natl Arts & Metiers, Inserm U944, CNRS UMR7212, Paris, France Biodim Mutabilis, F-93230 Romainville, France论文数: 引用数: h-index:机构:Emiliani, Stephane论文数: 0 引用数: 0 h-index: 0机构: Univ Paris 05, CNRS UMR 8104, Inserm U1016, Inst Cochin, F-75014 Paris, France Biodim Mutabilis, F-93230 Romainville, FranceRuff, Marc论文数: 0 引用数: 0 h-index: 0机构: Univ Strasbourg, CNRS, INSERM, IGBMC, F-67404 Illkirch Graffenstaden, France Biodim Mutabilis, F-93230 Romainville, FranceLedoussal, Benoit论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceMoreau, Francois论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, FranceBenarous, Richard论文数: 0 引用数: 0 h-index: 0机构: Biodim Mutabilis, F-93230 Romainville, France Biodim Mutabilis, F-93230 Romainville, France
- [47] A soluble active mutant of HIV-1 integrase - Involvement of both the core and carboxyl-terminal domains in multimerizationJOURNAL OF BIOLOGICAL CHEMISTRY, 1996, 271 (13) : 7712 - 7718Jenkins, TM论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892Engelman, A论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892Ghirlando, R论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892Craigie, R论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOLEC BIOL LAB,NIH,BETHESDA,MD 20892
- [48] Zinc folds the N-terminal domain of HIV-1 integrase, promotes multimerization, and enhances catalytic activityPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1996, 93 (24) : 13659 - 13664Zheng, RL论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOL BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOL BIOL LAB,NIH,BETHESDA,MD 20892Jenkins, TM论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOL BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOL BIOL LAB,NIH,BETHESDA,MD 20892Craigie, R论文数: 0 引用数: 0 h-index: 0机构: NIDDKD,MOL BIOL LAB,NIH,BETHESDA,MD 20892 NIDDKD,MOL BIOL LAB,NIH,BETHESDA,MD 20892
- [49] Inhibition of HIV-1 integrase nuclear import and replication by a peptide bearing integrase putative nuclear localization signalRETROVIROLOGY, 2009, 6Levin, Aviad论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, IsraelArmon-Omer, Ayelet论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel Ziv Med Ctr, IL-13100 Safed, Israel Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, IsraelRosenbluh, Joseph论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, IsraelMelamed-Book, Naomi论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, IsraelGraessmann, Adolf论文数: 0 引用数: 0 h-index: 0机构: Free Univ Berlin, Inst Mol Biol & Biochem, D-1000 Berlin, Germany Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, IsraelWaigmann, Elisabeth论文数: 0 引用数: 0 h-index: 0机构: Med Univ Vienna, Inst Med Biochem, Vienna Bioctr, Max Perutz Labs,Univ Dept, Vienna, Austria Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, IsraelLoyter, Abraham论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel
- [50] Peptides that inhibit HIV-1 integrase by blocking its protein-protein interactionsFEBS JOURNAL, 2012, 279 (16) : 2795 - 2809Maes, Michal论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Inst Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Inst Chem, IL-91904 Jerusalem, IsraelLoyter, Abraham论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Alexander Silberman Inst Life Sci, Dept Biol Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Inst Chem, IL-91904 Jerusalem, IsraelFriedler, Assaf论文数: 0 引用数: 0 h-index: 0机构: Hebrew Univ Jerusalem, Inst Chem, IL-91904 Jerusalem, Israel Hebrew Univ Jerusalem, Inst Chem, IL-91904 Jerusalem, Israel