Azacycloalkanes: XXXIX. New Syntheses of 1H-Pyrrole-1-carboxylic acid and 1,2-dihydropyrrolo-[1,2-a]pyrazin-3(4H)-one derivatives

被引：0
|
作者：
G. V. Mokrov
A. M. Likhosherstov
V. S. Troitskaya
T. A. Gudasheva
机构：
[1] Russian Academy of Medical Sciences,Zakusov Research Institute of Pharmacology
来源：
Russian Journal of Organic Chemistry | 2009年 / 45卷
关键词：
Pyrazin; Thionyl Chloride; Reductive Amination; Alkanoic Acid; Amino Ester;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
New procedures have been developed for the synthesis of α-(2-formyl-1H-pyrrol-1-yl)-substituted carboxylic acids, α-(2-R-aminomethyl-1H-pyrrol-1-yl)-substituted carboxylic acids, and 1,2-dihydropyrrolo-[1,2-a]pyrazin-3(4H)-ones on the basis of furfurol and α-amino acids.
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页码：1829 / 1833
页数：4
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