5-HT1A receptor blockade reverses GABAA receptor α3 subunit-mediated anxiolytic effects on stress-induced hyperthermia

被引:0
|
作者
Christiaan H. Vinkers
Ruud van Oorschot
S. Mechiel Korte
Berend Olivier
Lucianne Groenink
机构
[1] Utrecht University,Division of Pharmacology, Utrecht Institute for Pharmaceutical Sciences and Rudolf Magnus Institute of Neuroscience
[2] Yale University School of Medicine,Department of Psychiatry
来源
Psychopharmacology | 2010年 / 211卷
关键词
Interaction; Zolpidem; TP003; Benzodiazepine; Serotonin antagonist; Serotonergic; WAY-100635; WAY100,635; alpha3; alpha 3; Stress; Anxiety;
D O I
暂无
中图分类号
学科分类号
摘要
引用
收藏
页码:123 / 130
页数:7
相关论文
共 50 条
  • [21] SSRI exerts anxiolytic effect via amygdalar 5-HT1A receptor
    Izumi, Takeshi
    Wang, Ce
    Ohmura, Yu
    Yoshida, Takayuki
    Yoshioka, Mitsuhiro
    JOURNAL OF PHARMACOLOGICAL SCIENCES, 2016, 130 (03) : S122 - S122
  • [22] EFFECTS OF COLD STRESS ON SOME 5-HT1A, 5-HT1C AND 5-HT2 RECEPTOR-MEDIATED RESPONSES
    ZAMFIR, O
    BROQUA, P
    BAUDRIE, V
    CHAOULOFF, F
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1992, 219 (02) : 261 - 269
  • [23] The Gαi subunit links the 5-HT1A receptor to a GIRK
    Mueller, NK
    Beck, SG
    FASEB JOURNAL, 1999, 13 (04): : A134 - A134
  • [24] EFFECTS OF NOVEL 5-HT1A RECEPTOR ANTAGONISTS ON MEASURES OF POSTSYNAPTIC 5-HT1A RECEPTOR ACTIVATION IN-VIVO
    THIELEN, RJ
    FRAZER, A
    LIFE SCIENCES, 1995, 56 (07) : PL163 - PL168
  • [25] Juvenile stress-induced alteration of GABAA receptor alpha subunit maturation in the rat
    Jacobson-Pick, S
    Vender, S
    Elkobi, A
    Rosenblum, K
    Richter-Levin, G
    REVIEWS IN THE NEUROSCIENCES, 2005, 16 : S33 - S33
  • [26] 5-HT1A receptor knockout mice and anxiety: Is the GABAA-benzodiazepine receptor complex involved?
    Olivier, B
    Groenink, L
    Van der Gugten, J
    EUROPEAN NEUROPSYCHOPHARMACOLOGY, 2002, 12 : S153 - S154
  • [27] Role of 5-HT1A Receptor in the Anxiolytic-Relaxant Effects of Bergamot Essential Oil in Rodent
    Rombola, Laura
    Scuteri, Damiana
    Watanabe, Chizuko
    Sakurada, Shinobu
    Hamamura, Kengo
    Sakurada, Tsukasa
    Tonin, Paolo
    Corasaniti, Maria Tiziana
    Bagetta, Giacinto
    Morrone, Luigi Antonio
    INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2020, 21 (07)
  • [28] Effects of corticosterone on 5-HT1A and 5-HT2 receptor binding and on the receptor-mediated behavioral responses of rats
    Takao, K
    Nagatani, T
    Kitamura, Y
    Yamawaki, S
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1997, 333 (2-3) : 123 - 128
  • [29] 5-HT1A RECEPTOR BLOCKADE INCREASES PENILE ERECTIONS INDUCED BY INDIRECT SEROTONIN AGONISTS
    SIMON, P
    BERTRAND, J
    COSTENTIN, J
    NEUROREPORT, 1993, 5 (03) : 229 - 230
  • [30] 5-HT1A receptor and 5-HT1B receptor knockout mice in stress and anxiety paradigms
    Groenink, L
    van Bogaert, MJV
    van der Gugten, J
    Oosting, RS
    Olivier, B
    BEHAVIOURAL PHARMACOLOGY, 2003, 14 (5-6): : 369 - 383