Synthesis and structure of 3-(3-acetoxyalkylcarbamoyl-4-hydroxy-2-oxo-1,2-dihydroquinolin-1-yl)propanoic acids

被引：0
|
作者：
I. V. Ukrainets
O. V. Gorokhova
K. V. Andreeva
机构：
[1] National University of Pharmacy,
来源：
Russian Journal of Organic Chemistry | 2014年 / 50卷
关键词：
Propanoic Acid; Torsion Angle; AcOH; Colorless Crystal; Cyano Group;
D O I：
暂无
中图分类号：
学科分类号：
摘要：
Treatment of 1-(2-cyanoethyl)-4-hydroxy-N-(hydroxyalkyl)-2-oxo-1,2-dihydroquinoline-3-carboxamides with a solution of hydrogen chloride in aqueous acetic acid ensures selective transformation of the cyano group into amide or carboxy with simultaneous acetylation of the hydroxyalkyl fragments.
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页码：63 / 65
页数：2
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