One-Pot Assembly of Alkyl [(5-Amino-1H-pyrrol-2-yl)sulfanyl]-acetates from Propargylamines, Isothiocyanates, and Alkyl Bromoacetates

被引：0
|
作者：
O. A. Tarasova
N. A. Nedolya
B. A. Trofimov
机构：
[1] Russian Academy of Sciences,Favorskii Irkutsk Institute of Chemistry, Siberian Branch
来源：
Russian Journal of Organic Chemistry | 2018年 / 54卷
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摘要：
Methyl and tert-butyl 2-{[5-(diethylamino)-1-methyl-1H-pyrrol-2-yl]sulfanyl|acetates have been synthesized in one preparative stage from accessible N,N-diethylprop-2-yn-1-amine, methyl isothiocyanate, and methyl 2-bromoacetate.
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页码：1325 / 1328
页数：3
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