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- [21] Discovery of preclinical development candidate inhibitors of the mediator complex-associated kinases CDK8 and CDK19 and evaluation of their therapeutic potentialCANCER RESEARCH, 2016, 76Clarke, Paul论文数: 0 引用数: 0 h-index: 0Esdar, Christina论文数: 0 引用数: 0 h-index: 0Mallinger, Aurelie论文数: 0 引用数: 0 h-index: 0Schiemann, Kai论文数: 0 引用数: 0 h-index: 0Waalboer, Dennis论文数: 0 引用数: 0 h-index: 0Crumpler, Simon论文数: 0 引用数: 0 h-index: 0Rink, Christian论文数: 0 引用数: 0 h-index: 0Stieber, Frank论文数: 0 引用数: 0 h-index: 0Calderini, Michel论文数: 0 引用数: 0 h-index: 0Adeniji-Popoola, Olajumoke论文数: 0 引用数: 0 h-index: 0Ortiz-Ruiz, Maria-Jesus论文数: 0 引用数: 0 h-index: 0Samant, Rahul S.论文数: 0 引用数: 0 h-index: 0Czodrowski, Paul论文数: 0 引用数: 0 h-index: 0Musil, Djordje论文数: 0 引用数: 0 h-index: 0Schwarz, Daniel论文数: 0 引用数: 0 h-index: 0Schneider, Klaus论文数: 0 引用数: 0 h-index: 0Busch, Michael论文数: 0 引用数: 0 h-index: 0Stubbs, Mark论文数: 0 引用数: 0 h-index: 0Burke, Rosemary论文数: 0 引用数: 0 h-index: 0TePoele, Robert论文数: 0 引用数: 0 h-index: 0Gowan, Sharon论文数: 0 引用数: 0 h-index: 0Rohdich, Felix论文数: 0 引用数: 0 h-index: 0Raynaud, Florence论文数: 0 引用数: 0 h-index: 0Schneider, Richard论文数: 0 引用数: 0 h-index: 0Poeschke, Oliver论文数: 0 引用数: 0 h-index: 0Blaukat, Andree论文数: 0 引用数: 0 h-index: 0Urbahns, Klaus论文数: 0 引用数: 0 h-index: 0Workman, Paul论文数: 0 引用数: 0 h-index: 0Kaufmann, Wolfgang论文数: 0 引用数: 0 h-index: 0Simon, Stephanie论文数: 0 引用数: 0 h-index: 0Eccles, Suzanne A.论文数: 0 引用数: 0 h-index: 0Dale, Trevor论文数: 0 引用数: 0 h-index: 0Wienke, Dirk论文数: 0 引用数: 0 h-index: 0Blagg, Julian论文数: 0 引用数: 0 h-index: 0
- [22] Elucidation of the different roles of CDK8 and CDK19 in colorectal cancer (CRC) using CRISPR gene editing technologyCANCER RESEARCH, 2016, 76Ruiz, Maria J. Ortiz论文数: 0 引用数: 0 h-index: 0Popoola, Olajumoke论文数: 0 引用数: 0 h-index: 0Mallinger, Aurelie论文数: 0 引用数: 0 h-index: 0Gowan, Sharon论文数: 0 引用数: 0 h-index: 0Court, Will论文数: 0 引用数: 0 h-index: 0Box, Gary论文数: 0 引用数: 0 h-index: 0Valenti, Melanie论文数: 0 引用数: 0 h-index: 0Brandon, Alexis De Haven论文数: 0 引用数: 0 h-index: 0Te-Poele, Robert论文数: 0 引用数: 0 h-index: 0Workman, Paul论文数: 0 引用数: 0 h-index: 0Schiemann, Kai论文数: 0 引用数: 0 h-index: 0Esdar, Cristina论文数: 0 引用数: 0 h-index: 0Wienke, Dirk论文数: 0 引用数: 0 h-index: 0Blagg, Julian论文数: 0 引用数: 0 h-index: 0Clarke, Paul论文数: 0 引用数: 0 h-index: 0Eccles, Suzanne A.论文数: 0 引用数: 0 h-index: 0
- [23] Distinct roles for Mediator Cdk8 module subunits in Drosophila developmentEMBO JOURNAL, 2007, 26 (04): : 1045 - 1054Loncle, Nicolas论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, FranceBoube, Muriel论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, FranceJoulia, Laurent论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, FranceBoschiero, Claire论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, FranceWerner, Michel论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, FranceCribbs, David L.论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, FranceBourbon, Henri-Marc论文数: 0 引用数: 0 h-index: 0机构: Univ Toulouse 3, CNRS, Ctr Dev Biol, UMR5544, Toulouse 09, France
- [24] Discovery of Potent, Selective, and Orally Bioavailable Small-Molecule Modulators of the Mediator Complex-Associated Kinases CDK8 and CDK19JOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (03) : 1078 - 1101Mallinger, Aurelie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandSchiemann, Kai论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandRink, Christian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandStieber, Frank论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandCalderini, Michel论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandCrumpler, Simon论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandStubbs, Mark论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandAdeniji-Popoola, Olajumoke论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandPoeschke, Oliver论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandBusch, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandCzodrowski, Paul论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandMusil, Djordje论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandSchwarz, Daniel论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandOrtiz-Ruiz, Maria-Jesus论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandSchneider, Richard论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandThai, Ching论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandValenti, Melanie论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandBrandon, Alexis de Haven论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandBurke, Rosemary论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandWorkman, Paul论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandDale, Trevor论文数: 0 引用数: 0 h-index: 0机构: Cardiff Univ, Sch Biosci, Cardiff CF10 3AX, S Glam, Wales Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandWienke, Dirk论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandClarke, Paul A.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandEsdar, Christina论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandRaynaud, Florence I.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandEccles, Suzanne A.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandRohdich, Felix论文数: 0 引用数: 0 h-index: 0机构: Merck KGaA, D-64293 Darmstadt, Germany Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, EnglandBlagg, Julian论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England Inst Canc Res, Canc Res UK Canc Therapeut Unit, London SW7 3RP, England
- [25] Inhibition of Cdk8/Cdk19 Activity Promotes Treg Cell Differentiation and Suppresses Autoimmune DiseasesFRONTIERS IN IMMUNOLOGY, 2019, 10Guo, Zengli论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Microbiol & Immunol, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USAWang, Gang论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Microbiol & Immunol, Chapel Hill, NC 27599 USA Xuzhou Med Univ, Canc Inst, Xuzhou, Jiangsu, Peoples R China Xuzhou Med Univ, Affiliated Hosp, Ctr Clin Oncol, Xuzhou, Jiangsu, Peoples R China Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USALv, Yanfang论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Canc Inst, Xuzhou, Jiangsu, Peoples R China Xuzhou Med Univ, Affiliated Hosp, Ctr Clin Oncol, Xuzhou, Jiangsu, Peoples R China Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USAWan, Yisong Y.论文数: 0 引用数: 0 h-index: 0机构: Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Dept Microbiol & Immunol, Chapel Hill, NC 27599 USA Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USAZheng, Junnian论文数: 0 引用数: 0 h-index: 0机构: Xuzhou Med Univ, Canc Inst, Xuzhou, Jiangsu, Peoples R China Xuzhou Med Univ, Affiliated Hosp, Ctr Clin Oncol, Xuzhou, Jiangsu, Peoples R China Univ North Carolina Chapel Hill, Lineberger Comprehens Canc Ctr, Chapel Hill, NC 27599 USA
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