Parallel synthesis of polysubstituted tetrahydroquinolines

被引：73
|
作者：
Baudelle, R [1 ]
Melnyk, P [1 ]
Déprez, B [1 ]
Tartar, A [1 ]
机构：
[1] CEREP, F-59000 Lille, France
来源：
TETRAHEDRON | 1998年 / 54卷 / 16期
关键词：
D O I：
10.1016/S0040-4020(98)00140-9
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A three-component cycloaddition was used to prepare a library of polysubtituted tetrahydroquinolines. Reaction conditions were optimised and a large range of anilines, aldehydes and alkenes were tested. (C) 1998 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：4125 / 4140
页数：16
相关论文
共 50 条
  • [41] Efficient synthesis of polysubstituted acylguanidines and guanylureas
    Katritzky, AR
    Rogovoy, BV
    Cai, XH
    Kirichenko, N
    Kovalenko, KV
    JOURNAL OF ORGANIC CHEMISTRY, 2004, 69 (02): : 309 - 313
  • [42] Synthesis of polysubstituted 4-fluoroquinolinones
    Kiselyov, AS
    Piatnitski, EL
    Doody, J
    ORGANIC LETTERS, 2004, 6 (22) : 4061 - 4063
  • [43] Regioselective synthesis of polysubstituted pyrazoles and isoxazoles
    Katritzky, AR
    Wang, MY
    Zhang, SM
    Vonkov, AVV
    Steel, PJ
    JOURNAL OF ORGANIC CHEMISTRY, 2001, 66 (20): : 6787 - 6791
  • [44] Regiospecific synthesis of polysubstituted furans and their application in organic synthesis
    Wong, HNC
    PURE AND APPLIED CHEMISTRY, 1996, 68 (02) : 335 - 344
  • [45] Synthesis of polysubstituted-2-naphthols
    Juteau, H
    Gareau, Y
    Lachance, H
    TETRAHEDRON LETTERS, 2005, 46 (27) : 4547 - 4549
  • [46] Synthesis and receptor affinity of polysubstituted adenosines
    Vittori, S
    Camaioni, E
    Costanzi, S
    Volpini, R
    Klotz, KN
    Cristalli, G
    NUCLEOSIDES & NUCLEOTIDES, 1999, 18 (4-5): : 739 - 740
  • [47] Short and stereoselective synthesis of polysubstituted cyclohexanones
    Geirsson, JKF
    Arnadottir, L
    Jonsson, S
    TETRAHEDRON, 2004, 60 (41) : 9149 - 9153
  • [48] A General and Scalable Synthesis of Polysubstituted Indoles
    Tejedor, David
    Diana-Rivero, Raquel
    Garcia-Tellado, Fernando
    MOLECULES, 2020, 25 (23):
  • [49] A cycloaddition approach toward the synthesis of substituted indolines and tetrahydroquinolines
    Padwa, A
    Brodney, MA
    Liu, B
    Satake, K
    Wu, T
    JOURNAL OF ORGANIC CHEMISTRY, 1999, 64 (10): : 3595 - 3607
  • [50] Tandem synthesis of tetrahydroquinolines and identification of the reaction network byoperandoNMR
    Chen, Jingwen
    Qi, Long
    Zhang, Biying
    Chen, Minda
    Kobayashi, Takeshi
    Bao, Zongbi
    Yang, Qiwei
    Ren, Qilong
    Huang, Wenyu
    Zhang, Zhiguo
    Qi, Long (lqi@iastate.edu), 1600, Royal Society of Chemistry (11): : 4332 - 4341
12345