4-aryl-2,4-dioxobutanoic acid inhibitors of HIV-1 integrase and viral replication in cells

被引：221
|
作者：
Wai, JS
Egbertson, MS
Payne, LS
Fisher, TE
Embrey, MW
Tran, LO
Melamed, JY
Langford, HM
Guare, JP
Zhuang, LG
Grey, VE
Vacca, JP
Holloway, MK
Naylor-Olsen, AM
Hazuda, DJ
Felock, PJ
Wolfe, AL
Stillmock, KA
Schleif, WA
Gabryelski, LJ
Young, SD
机构：
[1] Merck Res Labs, Dept Med Chem, W Point, PA 19486 USA
[2] Merck Res Labs, Dept Mol Syst, W Point, PA 19486 USA
[3] Merck Res Labs, Dept Antiviral Res, W Point, PA 19486 USA
来源：
JOURNAL OF MEDICINAL CHEMISTRY | 2000年 / 43卷 / 26期
关键词：
D O I：
10.1021/jm000176b
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
引用
收藏
页码：4923 / 4926
页数：4
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