Bisclder-Napieralski synthesis of some new pyrazole-fused β-carbolines

被引:0
|
作者
Abu-Safieh, KA
El-Abadelah, MM
Sabri, SS
Voelter, W
Mössmer, CM
Stroebele, M
机构
[1] Univ Tubingen, Phys Biochem Abt, Inst Physiol Chem, D-72076 Tubingen, Germany
[2] Univ Jordan, Dept Chem, Fac Sci, Amman, Jordan
[3] Univ Tubingen, Inst Anorgan Chem, D-72076 Tubingen, Germany
关键词
Bischler-Napieralski reaction; directed cyclization; pyrazolopyridoindoles;
D O I
暂无
中图分类号
O61 [无机化学];
学科分类号
070301 ; 081704 ;
摘要
3-(4-Acylaminopyrazol-5-yl)-4-methylindoles (13a,b), under Bischler-Napieralski reaction conditions, undergo cyclization at the pyrrolic carbon-2 with ultimate formation of the corresponding pyrazolo[3,4:5',6']pyrido[3,4-b]indoles (14a,b) as evidenced by crystal structure analysis of 14a.
引用
收藏
页码:1327 / 1332
页数:6
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