Oleamide Analogues as Positive Allosteric Modulators of the Serotonin (5-HT) 5-HT2C and 5-HT2A Receptors

被引：0
|
作者：
Chen, Jianping
Wold, Eric
Garcia, Erik
Pazdrak, Konrad
Wild, Christopher
Mifflin, Randy
Chen, Halving
Anastasio, Noelle
Cunningham, Kathryn
Zhou, Jia
机构：
来源：
FASEB JOURNAL | 2021年 / 35卷
关键词：
D O I：
10.1096/fasebj.2021.35.S1.04080
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页数：2
相关论文
共 50 条
  • [21] Synthesis, affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors and structure-activity relationships of a series of cyproheptadine analogues
    Honrubia, MA
    Rodriguez, J
    Dominguez, R
    Lozoya, E
    Manaut, F
    Seijas, JA
    Villaverde, MC
    Calleja, JM
    Cadavid, MI
    Maayani, S
    Sanz, F
    Loza, MI
    CHEMICAL & PHARMACEUTICAL BULLETIN, 1997, 45 (05) : 842 - 848
  • [22] Involvement of 5-HT2A Receptors in the Serotonin (5-HT) Syndrome caused by Excessive 5-HT Efflux in Rat Brain
    Krishnamoorthy, Swapna
    Ma, Zhiyuan
    Zhang, Gongliang
    Wei, Jianning
    Auerbach, Sidney B.
    Tao, Rui
    BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY, 2010, 107 (04) : 830 - 841
  • [23] Activities of novel aryloxyalkylimidazolines on rat 5-HT2A and 5-HT2C receptors
    Siegel, BW
    Freedman, J
    Vaal, MJ
    Baron, BM
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1996, 296 (03) : 307 - 318
  • [24] Effect of 5-HT2A and 5-HT2C receptors on temporal discrimination by mice
    Halberstadt, Adam L.
    Sindhunata, Ivan S.
    Scheffers, Kees
    Flynn, Aaron D.
    Sharp, Richard F.
    Geyer, Mark A.
    Young, Jared W.
    NEUROPHARMACOLOGY, 2016, 107 : 364 - 375
  • [25] Physiological relevance of constitutive activity of 5-HT2A and 5-HT2C receptors
    Berg, KA
    Harvey, JA
    Spampinato, U
    Clarke, WP
    TRENDS IN PHARMACOLOGICAL SCIENCES, 2005, 26 (12) : 625 - 630
  • [26] Serotonin 5-HT2A and 5-HT2C receptors as potential targets for modulation of psychostimulant use and dependence
    Bubar, Marcy J.
    Cunningham, Kathryn A.
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2006, 6 (18) : 1971 - 1985
  • [27] Generation of anti-peptide antibodies against serotonin 5-HT2A and 5-HT2C receptors
    Backstrom, JR
    SandersBush, E
    JOURNAL OF NEUROSCIENCE METHODS, 1997, 77 (01) : 109 - 117
  • [28] Agonist properties of N,N-Dimethyltryptamine at serotonin 5-HT2A and 5-HT2C receptors
    Smith, RL
    Canton, H
    Barrett, RJ
    Sanders-Bush, E
    PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, 1998, 61 (03) : 323 - 330
  • [29] Pharmacological Evaluations of a Novel Chemical Series of Serotonin 5-HT2C Receptor (5-HT2CR) Positive Allosteric Modulators
    Anastasio, Noelle
    Wold, Eric
    Garcia, Erik
    Pazdrak, Konrad
    Chen, Jianping
    Wild, Christopher
    Zhou, Jia
    Cunningham, Kathryn
    NEUROPSYCHOPHARMACOLOGY, 2019, 44 (SUPPL 1) : 200 - 201
  • [30] 5-HT2A and 5-HT2C receptor stimulation are differentially involved in the cortical dopamine release in 5-HT2A and 5-HT2C genetic mutant mice
    Huang, M.
    Li, Z.
    Prus, A. J.
    Dai, J.
    Meltzer, H. Y.
    SCHIZOPHRENIA BULLETIN, 2007, 33 (02) : 317 - 318
12345