The synthesis of heterocyclic products via C-H activation has won impressive advances as a newly emerging synthetic strategy. Herein, the recent research advances in heterocycle synthesis employing 8-aminoquinoline directed C-H activation, either in the form of direct intramolecular C-H elaboration or domino reactions involving the C-H activation and other transformation-based annulation reactions are highlighted.
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China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Hou, Xinjiao
Wang, Run
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Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R China
Fudan Univ, Sch Pharm, Dept Med Chem, Shanghai 201203, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Wang, Run
Fang, Feifei
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Lingang Lab, Shanghai 200031, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Fang, Feifei
Qu, Zhiyan
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Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Qu, Zhiyan
Zhou, Jianhui
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Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Zhou, Jianhui
Yu, Ting
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Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Yu, Ting
Wang, Dechuan
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China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Wang, Dechuan
Liu, Hong
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China Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R China
Univ Chinese Acad Sci, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, Hangzhou 310024, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
Liu, Hong
Zhou, Yu
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Chinese Acad Sci, Shanghai Inst Mat Med, Drug Discovery & Dev Ctr, Shanghai 201203, Peoples R China
Univ Chinese Acad Sci, Hangzhou Inst Adv Study, Sch Pharmaceut Sci & Technol, Hangzhou 310024, Peoples R ChinaChina Pharmaceut Univ, Dept Med Chem, Nanjing 210009, Peoples R China
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Sun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R ChinaSun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R China
Li, Jun-Ming
Weng, Jiang
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Sun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R ChinaSun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R China
Weng, Jiang
Lu, Gui
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Sun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R China
Sun Yat Sen Univ, Inst Human Virol, Guangzhou 510080, Guangdong, Peoples R ChinaSun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R China
Lu, Gui
Chan, Albert S. C.
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Sun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R ChinaSun Yat Sen Univ, Sch Pharmaceut Sci, Inst Med Chem, Guangzhou 510006, Guangdong, Peoples R China