Synthesis and Spectral Characterization of 1,5-Naphthyridine Derivatives through Cross-Coupling Suzuki Reaction

被引：0
|
作者：
Mohammed, Shireen [1 ]
Maher, Khalid Ali [1 ]
机构：
[1] Univ Zakho, Fac Sci, Dept Chem, Duhok, Kir, Iraq
来源：
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2019年 / 29卷 / 02期
关键词：
1,5-Naphthyridine derivatives; Heteroaromatic boronic acids; Cross-coupling process; Suzuki reaction; Palladium catalyst; CYTOTOXICITY; AGENTS;
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The present work describes the synthesis of new 1,5-naphthyridine derivatives. The procedure is based on the cross-coupling reaction of commercially available 2-iodo-1,5-naphthyridine with aromatic and heteroaromatic boronic acids through the Suzuki reaction. This process furnished the desired products in high yields. The structures of all the new products obtained in this work are supported by spectral and analytical data. [GRAPHICS] .
引用
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页码：199 / 203
页数：5
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