Synthesis of 1,1-bis(1,2,4-triazol-1-yl)-based potential aromatase inhibitors

被引:1
|
作者
Katritzky, AR [1 ]
Pastor, A [1 ]
Voronkov, MV [1 ]
机构
[1] Univ Florida, Dept Chem, Ctr Heterocycl Cpds, Gainesville, FL 32611 USA
关键词
D O I
10.1002/jhet.5570370412
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Reactions of bis-(1,2,4-triazolyl) sulfoxide 2 with various carbonyl compounds 3 led to the formation of twelve corresponding I,1-bis-(1,2,4-triazolyl) compounds, with structures resembling closely some previously prepared aromatase inhibitors.
引用
收藏
页码:743 / 745
页数:3
相关论文
共 50 条
  • [1] SYNTHESIS OF 1-(1,2,4-TRIAZOL-1-YL)ETHYLBENZENE
    GOLUBIN, AI
    TIMOKHIN, BV
    ZINCHENKO, SV
    ZHURNAL ORGANICHESKOI KHIMII, 1993, 29 (11): : 2324 - 2325
  • [2] Synthesis, Crystal Structure and Luminescent Properties of 2D Zinc Coordination Polymers Based on Bis(1,2,4-triazol-1-yl)methane and 1,3-Bis(1,2,4-triazol-1-yl)propane
    Semitut, Evgeny
    Sukhikh, Taisiya
    Filatov, Evgeny
    Ryadun, Alexey
    Potapov, Andrei
    CRYSTALS, 2017, 7 (12):
  • [3] Azolyl derivatives of nitrohalobutadienes - II. Synthesis and certain reaction of 1,1-bis(3,5-dimethylpyrazol-1-yl)-2-nitrotrihalo-1,3-butadienes and 1,1-bis(1,2,4-triazol-1-yl)-2-nitrotrihalo-1,3-butadienes
    Zapolskii, VA
    Potkin, VI
    Nechai, NI
    Kaberdin, RV
    Pevzner, MS
    ZHURNAL ORGANICHESKOI KHIMII, 1997, 33 (11): : 1715 - 1720
  • [4] REARRANGEMENT OF (1,2,4-TRIAZOL-4-YL)ETHANOLS TO (1,2,4-TRIAZOL-1-YL)ETHANOLS
    BENTLEY, TW
    HOWLE, LM
    WAREHAM, PJ
    JONES, RVH
    TETRAHEDRON, 1992, 48 (37) : 7869 - 7878
  • [5] 4-(1,2,4-Triazol-1-yl)aniline
    Fun, Hoong-Kun
    Quah, Ching Kheng
    Chandrakantha, B.
    Isloor, Arun M.
    Shetty, Prakash
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2011, 67 : O164 - U2804
  • [6] 9-(1,2,4-Triazol-1-yl)anthracene
    Li, Rong
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2007, 63 : O2898 - U2403
  • [7] Molecular and crystal structures of bis{1,4-bis(1,2,4-triazol-1-yl)butane}dichlorocobalt(II)
    L. Shen
    Russian Journal of Coordination Chemistry, 2009, 35 : 772 - 775
  • [8] Molecular and crystal structures of bis{1,4-bis(1,2,4-triazol-1-yl)butane}dichlorocobalt(II)
    Shen, L.
    RUSSIAN JOURNAL OF COORDINATION CHEMISTRY, 2009, 35 (10) : 772 - 775
  • [9] Molecular and crystal structure of bis{1,4-bis(1,2,4-triazol-1-yl)butane}dibromocadmium(II)
    L. Shen
    Russian Journal of Coordination Chemistry, 2010, 36 : 117 - 119
  • [10] Photoluminescent Lanthanide(III) Coordination Polymers with Bis(1,2,4-Triazol-1-yl)Methane Linker
    Ivanova, Elizaveta A.
    Smirnova, Ksenia S.
    Pozdnyakov, Ivan P.
    Potapov, Andrei S.
    Lider, Elizaveta V.
    INORGANICS, 2023, 11 (08)