The preparation of 4,5-dihydro-3-aryl-naphth-[1,2-c]-isoxazoles from dilithiated 1-tetralone oxime and aromatic esters

被引：5

作者：

Beam, CF ^{[1
]}

Schady, DA ^{[1
]}

Rose, KL ^{[1
]}

Kelley, W ^{[1
]}

Rakkhit, R ^{[1
]}

Hornsby, CD ^{[1
]}

Studer-Martinez, SL ^{[1
]}

机构：

[1] Coll Charleston, Dept Chem & Biochem, Charleston, SC 29424 USA

来源：

SYNTHETIC COMMUNICATIONS | 2000年 / 30卷 / 18期

基金：

美国国家科学基金会;

关键词：

D O I：

10.1080/00397910008086979

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Dilithiated 1-tetralone oxime was prepared in excess lithium diisopropylamide and condensed with a variety of esters followed by acid cyclization of C-acylated intermediates to substituted 4,5-dihydronaphth-[1,2-c]isoxazoles.

引用

页码：3391 / 3404

页数：14

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