How blocking Raf activates the MAPK pathway

被引:3
|
作者
McCormick, Frank [1 ]
机构
[1] Univ Calif San Francisco, San Francisco, CA 94143 USA
关键词
KINASE; BRAF;
D O I
10.1111/j.1755-148X.2010.00680.x
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
引用
收藏
页码:187 / 189
页数:3
相关论文
共 50 条
  • [1] The Ras/Raf/MAPK pathway
    Molina, Julian R.
    Adjei, Alex A.
    JOURNAL OF THORACIC ONCOLOGY, 2006, 1 (01) : 7 - 9
  • [2] Allosteric activation of RAF in the MAPK signaling pathway
    Tsai, Chung-Jung
    Nussinov, Ruth
    CURRENT OPINION IN STRUCTURAL BIOLOGY, 2018, 53 : 100 - 106
  • [3] RAF inhibitors that evade paradoxical MAPK pathway activation
    Chao Zhang
    Wayne Spevak
    Ying Zhang
    Elizabeth A. Burton
    Yan Ma
    Gaston Habets
    Jiazhong Zhang
    Jack Lin
    Todd Ewing
    Bernice Matusow
    Garson Tsang
    Adhirai Marimuthu
    Hanna Cho
    Guoxian Wu
    Weiru Wang
    Daniel Fong
    Hoa Nguyen
    Songyuan Shi
    Patrick Womack
    Marika Nespi
    Rafe Shellooe
    Heidi Carias
    Ben Powell
    Emily Light
    Laura Sanftner
    Jason Walters
    James Tsai
    Brian L. West
    Gary Visor
    Hamid Rezaei
    Paul S. Lin
    Keith Nolop
    Prabha N. Ibrahim
    Peter Hirth
    Gideon Bollag
    Nature, 2015, 526 : 583 - 586
  • [4] RAF inhibitors that evade paradoxical MAPK pathway activation
    Zhang, Chao
    Spevak, Wayne
    Zhang, Ying
    Burton, Elizabeth A.
    Ma, Yan
    Habets, Gaston
    Zhang, Jiazhong
    Lin, Jack
    Ewing, Todd
    Matusow, Bernice
    Tsang, Garson
    Marimuthu, Adhirai
    Cho, Hanna
    Wu, Guoxian
    Wang, Weiru
    Fong, Daniel
    Hoa Nguyen
    Shi, Songyuan
    Womack, Patrick
    Nespi, Marika
    Shellooe, Rafe
    Carias, Heidi
    Powell, Ben
    Light, Emily
    Sanftner, Laura
    Walters, Jason
    Tsai, James
    West, Brian L.
    Visor, Gary
    Rezaei, Hamid
    Lin, Paul S.
    Nolop, Keith
    Ibrahim, Prabha N.
    Hirth, Peter
    Bollag, Gideon
    NATURE, 2015, 526 (7574) : 583 - U298
  • [5] BPTF activates the MAPK pathway through coexpression with Raf1 to promote proliferation of T-cell lymphoma
    Bai, Dongyu
    Zhou, Yong
    Shen, Fayan
    Gao, Dehong
    Suo, Wenhao
    Zhang, Haiping
    Li, Heng
    ONCOLOGY LETTERS, 2022, 24 (01)
  • [6] RAF inhibitors activate MAPK pathway through relief of RAF auto-inhibition
    Hoderfield, Matthew
    Merritt, Hanne
    Chan, John
    Wallroth, Marco
    Tandeske, Laura
    Hardy, Steve
    Hekmat-Nejad, Mohammad
    McCormick, Frank
    Nagel, Tobi
    CANCER RESEARCH, 2011, 71
  • [7] RAF Inhibitors Activate the MAPK Pathway by Relieving Inhibitory Autophosphorylation
    Holderfield, Matthew
    Merritt, Hanne
    Chan, John
    Wallroth, Marco
    Tandeske, Laura
    Zhai, Huili
    Tellew, John
    Hardy, Stephen
    Hekmat-Nejad, Mohammad
    Stuart, Darrin D.
    McCormick, Frank
    Nagel, Tobi E.
    CANCER CELL, 2013, 23 (05) : 594 - 602
  • [8] RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growth
    Georgia Hatzivassiliou
    Kyung Song
    Ivana Yen
    Barbara J. Brandhuber
    Daniel J. Anderson
    Ryan Alvarado
    Mary J. C. Ludlam
    David Stokoe
    Susan L. Gloor
    Guy Vigers
    Tony Morales
    Ignacio Aliagas
    Bonnie Liu
    Steve Sideris
    Klaus P. Hoeflich
    Bijay S. Jaiswal
    Somasekar Seshagiri
    Hartmut Koeppen
    Marcia Belvin
    Lori S. Friedman
    Shiva Malek
    Nature, 2010, 464 : 431 - 435
  • [9] RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growth
    Hatzivassiliou, Georgia
    Song, Kyung
    Yen, Ivana
    Brandhuber, Barbara J.
    Anderson, Daniel J.
    Alvarado, Ryan
    Ludlam, Mary J. C.
    Stokoe, David
    Gloor, Susan L.
    Vigers, Guy
    Morales, Tony
    Aliagas, Ignacio
    Liu, Bonnie
    Sideris, Steve
    Hoeflich, Klaus P.
    Jaiswal, Bijay S.
    Seshagiri, Somasekar
    Koeppen, Hartmut
    Belvin, Marcia
    Friedman, Lori S.
    Malek, Shiva
    NATURE, 2010, 464 (7287) : 431 - U132
  • [10] RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growth
    Hatzivassiliou, Georgia
    Song, Kyung
    Yen, Lvana
    Brandhuber, Barbara J.
    Anderson, Daniel J.
    Alvarado, Ryan
    Ludlam, Mary Jc
    Stokoe, David
    Gloor, Susan L.
    Vigers, Guy
    Morales, Tony
    Aliagas, Ignacio
    Liu, Bonnie
    Sideris, Steve
    Hoeflich, Klaus
    Jaiswal, Bijay S.
    Seshagiri, Sonnasekar
    Koeppen, Hartmut
    Belvin, Marcia
    Friedman, Lori S.
    Malek, Shiva
    CANCER RESEARCH, 2010, 70