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- [1] RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growthNature, 2010, 464 : 431 - 435Georgia Hatzivassiliou论文数: 0 引用数: 0 h-index: 0机构: Genentech,Kyung Song论文数: 0 引用数: 0 h-index: 0机构: Genentech,Ivana Yen论文数: 0 引用数: 0 h-index: 0机构: Genentech,Barbara J. Brandhuber论文数: 0 引用数: 0 h-index: 0机构: Genentech,Daniel J. Anderson论文数: 0 引用数: 0 h-index: 0机构: Genentech,Ryan Alvarado论文数: 0 引用数: 0 h-index: 0机构: Genentech,Mary J. C. Ludlam论文数: 0 引用数: 0 h-index: 0机构: Genentech,David Stokoe论文数: 0 引用数: 0 h-index: 0机构: Genentech,Susan L. Gloor论文数: 0 引用数: 0 h-index: 0机构: Genentech,Guy Vigers论文数: 0 引用数: 0 h-index: 0机构: Genentech,Tony Morales论文数: 0 引用数: 0 h-index: 0机构: Genentech,Ignacio Aliagas论文数: 0 引用数: 0 h-index: 0机构: Genentech,Bonnie Liu论文数: 0 引用数: 0 h-index: 0机构: Genentech,Steve Sideris论文数: 0 引用数: 0 h-index: 0机构: Genentech,Klaus P. Hoeflich论文数: 0 引用数: 0 h-index: 0机构: Genentech,Bijay S. Jaiswal论文数: 0 引用数: 0 h-index: 0机构: Genentech,Somasekar Seshagiri论文数: 0 引用数: 0 h-index: 0机构: Genentech,Hartmut Koeppen论文数: 0 引用数: 0 h-index: 0机构: Genentech,Marcia Belvin论文数: 0 引用数: 0 h-index: 0机构: Genentech,Lori S. Friedman论文数: 0 引用数: 0 h-index: 0机构: Genentech,Shiva Malek论文数: 0 引用数: 0 h-index: 0机构: Genentech,
- [2] RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growthNATURE, 2010, 464 (7287) : 431 - U132Hatzivassiliou, Georgia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASong, Kyung论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAYen, Ivana论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABrandhuber, Barbara J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Genentech Inc, San Francisco, CA 94080 USAAnderson, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAAlvarado, Ryan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALudlam, Mary J. C.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAStokoe, David论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAGloor, Susan L.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Genentech Inc, San Francisco, CA 94080 USAVigers, Guy论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Genentech Inc, San Francisco, CA 94080 USAMorales, Tony论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma, Boulder, CO 80301 USA Genentech Inc, San Francisco, CA 94080 USAAliagas, Ignacio论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALiu, Bonnie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASideris, Steve论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHoeflich, Klaus P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAJaiswal, Bijay S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASeshagiri, Somasekar论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAKoeppen, Hartmut论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABelvin, Marcia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAFriedman, Lori S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAMalek, Shiva论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [3] Registered report: RAF inhibitors prime wild-type RAF to activate the MAPK pathway and enhance growthELIFE, 2016, 5Bhargava, Ajay论文数: 0 引用数: 0 h-index: 0机构: Shakti BioRes, Woodbridge, NJ USA Shakti BioRes, Woodbridge, NJ USAPelech, Steven论文数: 0 引用数: 0 h-index: 0机构: Kinexus Bioinformat Corp, Vancouver, BC, Canada Shakti BioRes, Woodbridge, NJ USABen Woodard论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Biotechnol Res & Educ Program, College Pk, MD 20742 USA Shakti BioRes, Woodbridge, NJ USAKerwin, John论文数: 0 引用数: 0 h-index: 0机构: Univ Maryland, Biotechnol Res & Educ Program, College Pk, MD 20742 USA Shakti BioRes, Woodbridge, NJ USAMaherali, Nimet论文数: 0 引用数: 0 h-index: 0机构: Harvard Stem Cell Inst, Cambridge, MA USA Shakti BioRes, Woodbridge, NJ USA
- [4] RAF inhibitors activate MAPK pathway through relief of RAF auto-inhibitionCANCER RESEARCH, 2011, 71Hoderfield, Matthew论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAMerritt, Hanne论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAChan, John论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAWallroth, Marco论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USATandeske, Laura论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAHardy, Steve论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAHekmat-Nejad, Mohammad论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAMcCormick, Frank论文数: 0 引用数: 0 h-index: 0机构: UCSF Helen Diller Family, Ctr Comprehens Canc, San Francisco, CA USA Novartis Inst Biomed Res, Emeryville, CA USANagel, Tobi论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USA
- [5] RAF Inhibitors Activate the MAPK Pathway by Relieving Inhibitory AutophosphorylationCANCER CELL, 2013, 23 (05) : 594 - 602Holderfield, Matthew论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAMerritt, Hanne论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAChan, John论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAWallroth, Marco论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USATandeske, Laura论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAZhai, Huili论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Cambridge, MA 02139 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USATellew, John论文数: 0 引用数: 0 h-index: 0机构: Novartis Res Fdn, Genom Inst, San Diego, CA 92121 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAHardy, Stephen论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAHekmat-Nejad, Mohammad论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAStuart, Darrin D.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USAMcCormick, Frank论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, San Francisco, CA 94158 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USANagel, Tobi E.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA 94608 USA Novartis Inst Biomed Res, Emeryville, CA 94608 USA
- [6] RAF inhibitors transactivate RAF dimers and ERK signalling in cells with wild-type BRAFNATURE, 2010, 464 (7287) : 427 - U126Poulikakos, Poulikos I.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Dept Med, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USAZhang, Chao论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Howard Hughes Med Inst, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Cellular & Mol Pharmacol, San Francisco, CA 94158 USA Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USABollag, Gideon论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc, Berkeley, CA 94710 USA Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USAShokat, Kevan M.论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Howard Hughes Med Inst, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Cellular & Mol Pharmacol, San Francisco, CA 94158 USA Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USARosen, Neal论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Dept Med, New York, NY 10065 USA Mem Sloan Kettering Canc Ctr, Program Mol Pharmacol & Chem, New York, NY 10065 USA
- [7] RAF inhibitors transactivate RAF dimers and ERK signalling in cells with wild-type BRAFNature, 2010, 464 : 427 - 430Poulikos I. Poulikakos论文数: 0 引用数: 0 h-index: 0机构: Memorial Sloan-Kettering Cancer Center,Program in Molecular Pharmacology and Chemistry and Department of MedicineChao Zhang论文数: 0 引用数: 0 h-index: 0机构: Memorial Sloan-Kettering Cancer Center,Program in Molecular Pharmacology and Chemistry and Department of MedicineGideon Bollag论文数: 0 引用数: 0 h-index: 0机构: Memorial Sloan-Kettering Cancer Center,Program in Molecular Pharmacology and Chemistry and Department of MedicineKevan M. Shokat论文数: 0 引用数: 0 h-index: 0机构: Memorial Sloan-Kettering Cancer Center,Program in Molecular Pharmacology and Chemistry and Department of MedicineNeal Rosen论文数: 0 引用数: 0 h-index: 0机构: Memorial Sloan-Kettering Cancer Center,Program in Molecular Pharmacology and Chemistry and Department of Medicine
- [8] RAF inhibitors transactivate RAF dimers and ERK signaling in a wild-type BRAF-dependent mannerCANCER RESEARCH, 2010, 70Poulikakos, Poulikos I.论文数: 0 引用数: 0 h-index: 0Zhang, Chao论文数: 0 引用数: 0 h-index: 0Joseph, Eric W.论文数: 0 引用数: 0 h-index: 0Persaud, Yogindra论文数: 0 引用数: 0 h-index: 0Pratilas, Christine A.论文数: 0 引用数: 0 h-index: 0Bollag, Gideon论文数: 0 引用数: 0 h-index: 0Solit, David B.论文数: 0 引用数: 0 h-index: 0Shokat, Kevan M.论文数: 0 引用数: 0 h-index: 0Rosen, Neal论文数: 0 引用数: 0 h-index: 0
- [9] Wild-type and mutant B-RAF activate C-RAF through distinct mechanisms involving heterodimerizationMOLECULAR CELL, 2005, 20 (06) : 963 - 969Garnett, MJ论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Signal Transduct Team, Canc Res UK, Ctr Cell & Mol Biol, London SW3 6JB, EnglandRana, S论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Signal Transduct Team, Canc Res UK, Ctr Cell & Mol Biol, London SW3 6JB, EnglandPaterson, H论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Signal Transduct Team, Canc Res UK, Ctr Cell & Mol Biol, London SW3 6JB, EnglandBarford, D论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Signal Transduct Team, Canc Res UK, Ctr Cell & Mol Biol, London SW3 6JB, EnglandMarais, R论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res, Signal Transduct Team, Canc Res UK, Ctr Cell & Mol Biol, London SW3 6JB, England
- [10] RAF inhibitors that evade paradoxical MAPK pathway activationNature, 2015, 526 : 583 - 586Chao Zhang论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Wayne Spevak论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Ying Zhang论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Elizabeth A. Burton论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Yan Ma论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Gaston Habets论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Jiazhong Zhang论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Jack Lin论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Todd Ewing论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Bernice Matusow论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Garson Tsang论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Adhirai Marimuthu论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Hanna Cho论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Guoxian Wu论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Weiru Wang论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Daniel Fong论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Hoa Nguyen论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Songyuan Shi论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Patrick Womack论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Marika Nespi论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Rafe Shellooe论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Heidi Carias论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Ben Powell论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Emily Light论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Laura Sanftner论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Jason Walters论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,James Tsai论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Brian L. West论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Gary Visor论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Hamid Rezaei论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Paul S. Lin论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Keith Nolop论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Prabha N. Ibrahim论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Peter Hirth论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,Gideon Bollag论文数: 0 引用数: 0 h-index: 0机构: Plexxikon Inc.,