共 50 条
- [21] Design, synthesis and structure-activity relationships of 5-alkylaminoquinolines: Potent, orally active corticotropin-releasing factor-1 receptor antagonists[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 247Takeda, KunitoshiTerauchi, TaroHashizume, MinakoShikata, KohdohTaguchi, RyotaMurata-Tai, KaoruFujisawa, MasaeTakahashi, YoshinoriShin, KogyokuIno, MitsuhiroShibata, HisashiYonaga, Masahiro
- [22] Design and synthesis of a novel, achiral class of highly potent and selective, orally active neurokinin-1 receptor antagonists[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (05) : 1362 - 1365Hoffmann, TBös, MStadler, HSchnider, PHunkeler, WGodel, TGalley, GBallard, TMHiggins, GAPoli, SMSleight, AJ
- [23] Potent and selective, orally active adenosine A2A antagonists[J]. PURINERGIC SIGNALLING, 2012, 8 (01) : 124 - 125Flohr, A.Alanine, A.Moreau, J-LPoli, S.Riemer, C.
- [24] Design, synthesis and structure-activity relationships of novel uracil compounds as potent GNRH receptor antagonists.[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 223 : B137 - B137Zhu, YFStruthers, SSaunders, JGao, YHGross, TConnors, PReinhart, GLing, NChen, C
- [25] Discovery and structure-activity relationships of a novel series of fused piperidines as potent TRPM8 antagonists[J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 244Tamayo, Nuria
- [26] Design, synthesis, and structure-activity relationships of phthalimide-phenylpiperazines:: A novel series of potent and selective α1a-adrenergic receptor antagonists[J]. JOURNAL OF MEDICINAL CHEMISTRY, 2000, 43 (11) : 2183 - 2195Kuo, GHProuty, CMurray, WVPulito, VJolliffe, LCheung, PVarga, SEvangelisto, MWang, J
- [27] Pyrazolo Derivatives as Potent Adenosine Receptor Antagonists: An Overview on the Structure-Activity Relationships[J]. INTERNATIONAL JOURNAL OF MEDICINAL CHEMISTRY, 2011, 2011Cheong, Siew LeeVenkatesan, GopalakrishnanPaira, PriyankarJothibasu, RamasamyMandel, Alexander LaurenceFederico, StephanieSpalluto, GiampieroPastorin, Giorgia
- [28] Structure-activity relationships of thiazole and thiadiazole derivatives as potent and selective human adenosine A3 receptor antagonists[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2004, 12 (03) : 613 - 623Jung, KYKim, SKGao, ZGGross, ASMelman, NJacobson, KAKim, YC
- [29] Design, synthesis, and structure-activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists (vol 22, pg 6071, 2014)[J]. BIOORGANIC & MEDICINAL CHEMISTRY, 2015, 23 (13) : 3870 - 3870Yoshida, YuTerauchi, TaroNaoe, YoshimitsuKazuta, YujiOzaki, FumihiroBeuckmann, Carsten T.Nakagawa, MakotoSuzuki, MichiyukiKushida, IkuoTakenaka, OsamuUeno, TakashiYonaga, Masahiro
- [30] Structure-activity relationships and pharmacokinetic parameters of quinoline acylsulfonamides as potent and selective antagonists of the EP4 receptor[J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (06) : 2048 - 2054Burch, Jason D.Belley, MichelFortin, RejeanDeschenes, DenisGirard, MarioColucci, JohnFarand, JulieTherien, Alex G.Mathieu, Marie-ClaudeDenis, DanielleVigneault, ErikaLevesque, Jean-FrancoisGagne, SebastienWrona, MarkXu, DiagenClark, PatsyRowland, SteveHan, Yongxin