Green Suzuki coupling reaction for synthesis of abiraterone acetate and its analogues

被引：4
|
作者：
Bian, Xiaoqin [1 ,2 ]
Wang, Lizhong [2 ]
Liu, Jinliang [1 ]
Wang, Cunde [1 ]
机构：
[1] Yangzhou Univ, Sch Chem & Chem Engn, Yangzhou 225002, Jiangsu, Peoples R China
[2] Taizhou Polytech Coll, Sch Pharm, Taizhou 225300, Peoples R China
来源：
JOURNAL OF CHEMICAL RESEARCH | 2016年 / 05期
基金：
中国国家自然科学基金;
关键词：
abiraterone acetate; dehydroepiandrosterone; green Suzuki reaction; PEG-400; arylboronic acid; ORGANIC-SYNTHESIS; ROOM-TEMPERATURE; HIGHLY EFFICIENT; CATALYST-FREE; ON-WATER; AGENTS; WATER-PEG-400; HETEROCYCLES; DERIVATIVES; CHEMISTRY;
D O I：
10.3184/174751916X14604710386405
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
An eco-friendly efficient method was developed for the synthesis of abiraterone acetate and analogues in water-PEG-400 (6:1; v/v) at 75 degrees C from various arylboronic acids and 17-(trifluoromethanesulfonyl)oxy-3 beta-acetoxylandrosta-5,16-diene obtained from the 3-acetate of dehydroepiandrosterone.
引用
收藏
页码：289 / 292
页数：4
相关论文
共 50 条
  • [31] Synthesis of Au/Pd bimetallic nanoparticles and their application in the Suzuki coupling reaction
    Nasrollahzadeh, Mahmoud
    Azarian, Abbas
    Maham, Mehdi
    Ehsani, Ali
    [J]. JOURNAL OF INDUSTRIAL AND ENGINEERING CHEMISTRY, 2015, 21 : 746 - 748
  • [32] Ultrasound-assisted Suzuki coupling reaction for rapid synthesis of polydihexylfluorene
    Gao, Xu
    Lu, Ping
    Ma, Yuguang
    [J]. POLYMER, 2014, 55 (14) : 3083 - 3086
  • [33] Synthesis of novel dodecasubstituted porphyrins via the Suzuki coupling reaction.
    Muzzi, CM
    Medforth, CJ
    Smith, KM
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1997, 213 : 8 - ORGN
  • [34] A Concise Synthesis of (-)-Incrustoporin and its Analogues by Pd-catalyzed Suzuki-Miyaura Coupling from γ-Vinyl-γ-butyrolactone
    Nallasivam, Jothi L.
    Fernandes, Rodney A.
    [J]. CHEMISTRYSELECT, 2016, 1 (16): : 5137 - 5140
  • [35] Discovering Green, Aqueous Suzuki Coupling Reactions: Synthesis of Ethyl (4-Phenylphenyl)acetate, a Biaryl with Anti-Arthritic Potential
    Costa, Nancy E.
    Pelotte, Andrea L.
    Simard, Joseph M.
    Syvinski, Christopher A.
    Deveau, Amy M.
    [J]. JOURNAL OF CHEMICAL EDUCATION, 2012, 89 (08) : 1064 - 1067
  • [36] Efficient convergent synthesis of 1α,25-dihydroxyvitamin D3 and its analogues by Suzuki-Miyaura coupling
    Hanazawa, T
    Koyama, A
    Wada, T
    Morishige, E
    Okamoto, S
    Sato, F
    [J]. ORGANIC LETTERS, 2003, 5 (04) : 523 - 525
  • [37] Abiraterone-acetate/enzalutamideHypersensitivity reaction: case report
    [J]. Reactions Weekly, 2023, 1956 (1) : 14 - 14
  • [38] Green Suzuki-Miyaura cross-coupling for the synthesis of chiral biaryls
    Dotsenko, Irina A.
    Shishkina, Irina N.
    Demyanovich, Valeria M.
    Bumagin, Nikolay A.
    [J]. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 245
  • [39] Electrochemical synthesis and characterization of palladium nanoparticles on nafion-graphene support and its application for Suzuki coupling reaction
    Shendage, Suresh S.
    Patil, Umakant B.
    Nagarkar, Jayashree M.
    [J]. TETRAHEDRON LETTERS, 2013, 54 (26) : 3457 - 3461
  • [40] Synthesis of a palladium complex bearing 2-phenylbenzothiazole and its application to Suzuki-Miyaura coupling reaction
    Kosuru, Someswara Rao
    Lai, Hsin-Yu
    Yang, Chien-Yi
    Senadi, Gopal Chandru
    Lai, Yi-Chun
    Chen, Hsuan-Ying
    [J]. JOURNAL OF THE CHINESE CHEMICAL SOCIETY, 2019, 66 (01) : 110 - 113
12345