Green Suzuki coupling reaction for synthesis of abiraterone acetate and its analogues

被引：4
|
作者：
Bian, Xiaoqin [1 ,2 ]
Wang, Lizhong [2 ]
Liu, Jinliang [1 ]
Wang, Cunde [1 ]
机构：
[1] Yangzhou Univ, Sch Chem & Chem Engn, Yangzhou 225002, Jiangsu, Peoples R China
[2] Taizhou Polytech Coll, Sch Pharm, Taizhou 225300, Peoples R China
来源：
JOURNAL OF CHEMICAL RESEARCH | 2016年 / 05期
基金：
中国国家自然科学基金;
关键词：
abiraterone acetate; dehydroepiandrosterone; green Suzuki reaction; PEG-400; arylboronic acid; ORGANIC-SYNTHESIS; ROOM-TEMPERATURE; HIGHLY EFFICIENT; CATALYST-FREE; ON-WATER; AGENTS; WATER-PEG-400; HETEROCYCLES; DERIVATIVES; CHEMISTRY;
D O I：
10.3184/174751916X14604710386405
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
An eco-friendly efficient method was developed for the synthesis of abiraterone acetate and analogues in water-PEG-400 (6:1; v/v) at 75 degrees C from various arylboronic acids and 17-(trifluoromethanesulfonyl)oxy-3 beta-acetoxylandrosta-5,16-diene obtained from the 3-acetate of dehydroepiandrosterone.
引用
收藏
页码：289 / 292
页数：4
相关论文
共 50 条
  • [1] Efficient synthesis of isoflavone analogues via a Suzuki coupling reaction
    Ding, K
    Wang, SM
    [J]. TETRAHEDRON LETTERS, 2005, 46 (21) : 3707 - 3709
  • [2] Green synthesis of Pd nanoparticles supported on LDHs and its application in the Suzuki coupling reaction
    Liu, G. H.
    Bai, X. F.
    [J]. 2ND INTERNATIONAL CONFERENCE ON NEW MATERIAL AND CHEMICAL INDUSTRY (NMCI2017), 2018, 292
  • [3] The Suzuki coupling reaction in the stereocontrolled synthesis of 9-cis-retinoic acid and its ring-demethylated analogues
    Pazos, Y
    Iglesias, B
    de Lera, AR
    [J]. JOURNAL OF ORGANIC CHEMISTRY, 2001, 66 (25): : 8483 - 8489
  • [4] Green synthesis of novel chalcone and coumarin derivatives via Suzuki coupling reaction
    Vieira, Lucas C. C.
    Paixao, Marcio Weber
    Correa, Arlene G.
    [J]. TETRAHEDRON LETTERS, 2012, 53 (22) : 2715 - 2718
  • [5] Synthesis of Phenanthridines and Analogues via Suzuki Coupling and Condensation
    Dhara, Shubhendu
    Ghosh, Munmun
    Ray, Jayanta K.
    [J]. SYNLETT, 2013, 24 (17) : 2263 - 2265
  • [6] Synthesis of the marine sponge alkaloid oroidin and its analogues via Suzuki cross-coupling reactions
    Berrée, F
    Girard-Le Bleis, P
    Carboni, B
    [J]. TETRAHEDRON LETTERS, 2002, 43 (28) : 4935 - 4938
  • [7] Suzuki coupling based synthesis and in vitro cytotoxic evaluation of Fingolimod and analogues
    Mei, Tie-Wen
    Luo, Yu
    Feng, Xiang-Jun
    Lu, Wei
    Yang, Bo
    [J]. TETRAHEDRON, 2013, 69 (14) : 2927 - 2932
  • [8] Efficient synthesis of substituted terphenyls by suzuki coupling reaction
    Chaumeil, H
    Le Drian, C
    Defoin, A
    [J]. SYNTHESIS-STUTTGART, 2002, (06): : 757 - 760
  • [9] Synthesis of ditopic oligopyridines using the Suzuki coupling reaction
    Sielemann, D
    Winter, A
    Risch, N
    [J]. HETEROCYCLES, 2005, 65 (07) : 1663 - 1672
  • [10] Selective and efficient synthesis of decahedral palladium nanoparticles and its catalytic performance for Suzuki coupling reaction
    Patil, Aniruddha B.
    Patil, Dinkar S.
    Bhanage, Bhalchandra M.
    [J]. JOURNAL OF MOLECULAR CATALYSIS A-CHEMICAL, 2012, 365 : 146 - 153
12345