Synthesis of substituted 2-mercaptobenzaldehydes and 2-substituted benzo[b]thiophenes

被引：32
|
作者：
Gallagher, T
Pardoe, DA
Porter, RA
机构：
[1] Univ Bristol, Sch Chem, Bristol BS8 1TS, Avon, England
[2] SB Pharmaceut, Discovery Res, Harlow CM19 5AW, Essex, England
来源：
TETRAHEDRON LETTERS | 2000年 / 41卷 / 28期
关键词：
D O I：
10.1016/S0040-4039(00)00870-4
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Simple and rapid single-pot preparations of substituted 2-mercaptobenzaldehydes 5 and 2-substituted benzo[b]thiophenes 3 based on ortho-lithiation methodology are described. (C) 2000 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：5415 / 5418
页数：4
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