10-Camphorsulfonic acid ((±)-CSA) catalyzed facile one-pot synthesis of a new class of 2,5-disubstituted 1,3,4-oxadiazoles

被引：11

作者：

Mule, Siva Nagi Reddy ^{[1
,3
]}

Battula, Sailaja Kumari ^{[1
,3
]}

Velupula, Ganapathi ^{[1
]}

Guda, Dinneswara Reddy ^{[2
,4
]}

Bollikolla, Hari Babu ^{[1
]}

机构：

[1] Acharya Nagarjuna Univ, Dept Chem, Guntur 522510, Andhra Pradesh, India

[2] Yonsei Univ, Dept Chem & Med Chem, Wonju 220710, Gangwon Do, South Korea

[3] Hetero Res Fdn, APIE, Hyderabad 500018, Andhra Pradesh, India

[4] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India

来源：

RSC ADVANCES | 2014年 / 4卷 / 102期

关键词：

DERIVATIVES; ANTIBACTERIAL; CHEMISTRY;

D O I：

10.1039/c4ra11218k

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A convenient and efficient one-pot synthesis of 2,5-disubstituted-1,3,4-oxadizoles is described. Various carboxylic acid hydrazides reacted efficiently with different carboxylic acid chlorides and 10-camphorsulfonic acid. This methodology was successfully applied to the synthesis of a series of 2H-chromene substituted 1,3,4-oxadiazole derivatives in good to high yields.

引用

页码：58397 / 58403

页数：7

共 50 条

[21] A NEW EFFICIENT ONE-POT SYNTHESIS OF 2,5-DIARYL-1,3,4-OXADIAZOLES
Chiriac, Constantin I.
Tanasa, Fulga
Nechifor, Marioara
[J]. REVUE ROUMAINE DE CHIMIE, 2011, 56 (12) : 1113 - +
[22] Synthesis of 2,5-disubstituted 1,3,4-oxadiazoles as biologically active heterocycles
Kagthara, PR
Shah, NS
Doshi, RK
Parekh, HH
[J]. INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY, 1999, 38 (05): : 572 - 576
[23] Synthesis of 2,5-disubstituted 1,3,4-oxadiazoles containing benzothiazolylthiol grouping
Kelarev V.I.
Silin M.A.
Grigor'eva N.A.
Koshelev V.N.
[J]. Chemistry of Heterocyclic Compounds, 2000, 36 (2) : 207 - 213
[24] One-pot synthesis,antibacterial and antifungal activities of novel 2,5-disubstituted-1,3,4-oxadiazoles
Abdul Rauf
Shweta Sharma
Saloni Gangal
[J]. Chinese Chemical Letters, 2008, (01) : 5 - 8
[25] One-pot synthesis, antibacterial and antifungal activities of novel 2,5-disubstituted-1,3,4-oxadiazoles
Rauf, Abdul
Sharma, Shweta
Gangal, Saloni
[J]. CHINESE CHEMICAL LETTERS, 2008, 19 (01) : 5 - 8
[26] Synthesis of 2,5-disubstituted 1,3,4-oxadiazoles as potential antimicrobial agents
Undavia, NK
Trivedi, PB
Shanishchara, AP
Trivedi, VP
[J]. JOURNAL OF THE INDIAN CHEMICAL SOCIETY, 2005, 82 (08) : 746 - 747
[27] 2,5-DISUBSTITUTED 1,3,4-OXADIAZOLES - SYNTHESIS AND PRELIMINARY PHARMACOLOGICAL INVESTIGATION
MAZZONE, G
BONINA, F
PUGLISI, G
PANICO, AM
REINA, RA
[J]. FARMACO-EDIZIONE SCIENTIFICA, 1984, 39 (05): : 414 - 420
[28] Synthesis of 2,5-disubstituted 1,3,4-oxadiazoles using dry media
Kidwai, M
Mohan, R
[J]. ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL, 2003, 35 (04) : 426 - 429
[29] An expeditious and convenient one pot synthesis of 2,5-disubstituted-1,3,4-oxadiazoles
Mashraqui, SH
Ghadigaonkar, SG
Kenny, RS
[J]. SYNTHETIC COMMUNICATIONS, 2003, 33 (14) : 2541 - 2545
[30] A FACILE PROCEDURE FOR SYNTHESIS OF 2,5-DISUBSTITUTED-1,3,4-OXADIAZOLES
VAKULA, TR
SARASWAT.TV
SRINIVAS.VR
[J]. INDIAN JOURNAL OF CHEMISTRY, 1968, 6 (03): : 172 - &

← 1 2 3 4 5 →