Synthesis of Ugi-4CR boronate analogues via microwave irradiation

被引：2

作者：

Hsiao, Chao-Yu ^{[1
]}

Huang, Shi-Qing ^{[1
]}

Lien, Wan-Hsing ^{[1
]}

Hsu, Chen-Yun ^{[1
]}

Hsieh, Kun-lin ^{[1
]}

Lin, Meng-Hsuan ^{[1
]}

Wu, Meng-Ju ^{[1
]}

Fu, Chia-Chieh ^{[1
]}

Chen, Hsien-Chi ^{[1
]}

Fang, Hao-Ping ^{[1
]}

Li, Chia-Jung ^{[1
]}

Pan, Po-Shen ^{[1
]}

机构：

[1] Tamkang Univ, Dept Chem, 151 Yingzhuan Rd, New Taipei 25137, Taiwan

来源：

RESEARCH ON CHEMICAL INTERMEDIATES | 2017年 / 43卷 / 06期

关键词：

Boron; Multicomponent reaction; Ugi reaction; Suzuki-Miyaura cross-coupling; PEPTIDASE-4 INHIBITOR PHX1149; FACTOR-KAPPA-B; MULTICOMPONENT REACTIONS; PS-341;

D O I：

10.1007/s11164-016-2433-y

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The synthetic condition for the synthesis of boronate ester Ugi-4CR analogs under mild conditions was developed. The reported reactions were carried out in methanol and promoted by microwave heating. This synthetic strategy could provide unique access to a broad range of boron-containing chemical libraries.

引用

页码：3585 / 3597

页数：13

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