Three-component 2-aryl substituted benzothiophene formation under transition-metal free conditions

被引：21
|
作者：
Jiang, Pengcheng [1 ]
Che, Xingzong [1 ]
Liao, Yunfeng [1 ]
Huang, Huawen [1 ]
Deng, Guo-Jun [1 ]
机构：
[1] Xiangtan Univ, Coll Chem, Minist Educ, Key Lab Environm Friendly Chem & Applicat, Xiangtan 411105, Peoples R China
来源：
RSC ADVANCES | 2016年 / 6卷 / 48期
基金：
中国国家自然科学基金;
关键词：
C-H HETEROARYLATION; CARBOXYLIC-ACIDS; GENERAL-METHOD; DERIVATIVES; ACCESS; ARYLATION; CATALYST; RHODIUM; POTENT;
D O I：
10.1039/c6ra07730g
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A base-mediated 2-aryl substituted benzothiophene formation from 2-bromobenzene aldehydes, benzylic esters and elemental sulfur under transition-metal-free conditions is described. Various 2-aryl substituted benzothiophene were efficiently obtained under mild conditions.
引用
收藏
页码：41751 / 41754
页数：4
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