Effects of simvastatin on agonist-induced and GRK2-mediated β-adrenoceptor down-regulation in adult rat cardiomyocytes

被引:0
|
作者
Leineweber, K
Altmann, C
Harms, P
Brodde, OE
机构
[1] Univ Essen Gesamthsch Klinikum, Inst Pathophysiol, D-45122 Essen, Germany
[2] Univ Essen Gesamthsch Klinikum, Inst Pharmakol, D-45122 Essen, Germany
关键词
D O I
暂无
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
96
引用
收藏
页码:R27 / R27
页数:1
相关论文
共 50 条
  • [21] Agonist-induced Down-regulation of Endogenous Protein Kinase C α through an Endolysosomal Mechanism
    Lum, Michelle A.
    Pundt, Krista E.
    Paluch, Benjamin E.
    Black, Adrian R.
    Black, Jennifer D.
    [J]. JOURNAL OF BIOLOGICAL CHEMISTRY, 2013, 288 (18) : 13093 - 13109
  • [22] Effects of verapamil on down-regulation of norepinephrine-induced β adrenoceptors in cultured rat cardiomyocytes.
    Xu, B
    Zhang, SL
    Chen, RX
    [J]. ACTA PHARMACOLOGICA SINICA, 1998, 19 (02): : 148 - 150
  • [23] BETA-3-ADRENOCEPTOR AGONIST-INDUCED DOWN-REGULATION OF G(S)ALPHA AND FUNCTIONAL DESENSITIZATION IN A CHINESE-HAMSTER OVARY CELL-LINE EXPRESSING A BETA-3-ADRENOCEPTOR REFRACTORY TO DOWN-REGULATION
    CHAMBERS, J
    PARK, J
    CRONK, D
    CHAPMAN, C
    KENNEDY, FR
    WILSON, S
    MILLIGAN, G
    [J]. BIOCHEMICAL JOURNAL, 1994, 303 : 973 - 978
  • [24] CHARACTERIZATION AND AGONIST-INDUCED DOWN-REGULATION OF PARATHYROID-HORMONE RECEPTORS IN CLONAL RAT OSTEO-SARCOMA CELLS
    YAMAMOTO, I
    SHIGENO, C
    POTTS, JT
    SEGRE, GV
    [J]. ENDOCRINOLOGY, 1988, 122 (04) : 1208 - 1217
  • [25] DOWN-REGULATION OF CENTRAL RECEPTORS FOR THYROTROPIN-RELEASING-HORMONE IN KAPPA-OPIATE AGONIST-INDUCED ABSTINENCE IN THE RAT
    BHARGAVA, HN
    GULATI, A
    RAHMANI, NH
    [J]. NEUROPHARMACOLOGY, 1992, 31 (02) : 137 - 141
  • [26] Chronic clorgyline induces selective down-regulation of α2-adrenoceptor agonist binding sites in rat brain
    Miralles, A
    Ribas, C
    Escribá, PV
    García-Sevilla, JA
    [J]. PHARMACOLOGY & TOXICOLOGY, 2000, 87 (06): : 269 - 275
  • [27] Role of the rate of internalization of the agonist-receptor complex on the agonist-induced down-regulation of the lutropin/choriogonadotropin receptor
    Nakamura, K
    Lazari, MDM
    Li, SH
    Korgaonkar, C
    Ascoli, M
    [J]. MOLECULAR ENDOCRINOLOGY, 1999, 13 (08) : 1295 - 1304
  • [28] Taxol normalizes the impaired agonist-induced β2-adrenoceptor internalization in splenocytes from GRK2± mice
    Vroon, Anne
    Lombardi, Maria Stella
    Kavelaars, Annemieke
    Heijnen, Cobi J.
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 2007, 560 (01) : 9 - 16
  • [29] EVIDENCE FOR CELL TYPE DEPENDENT MECHANISMS IN AGONIST-INDUCED DOWN-REGULATION OF BETA-ADRENOCEPTORS
    RADEMAKER, B
    KRAMER, K
    BAST, A
    TIMMERMAN, H
    [J]. RESEARCH COMMUNICATIONS IN CHEMICAL PATHOLOGY AND PHARMACOLOGY, 1990, 67 (03): : 321 - 336
  • [30] Involvement of G protein-coupled receptor kinase (GRK) 3 and GRK2 in down-regulation of the α2B-adrenoceptor
    Desai, Aarti N.
    Salim, Samina
    Standifer, Kelly M.
    Eikenburg, Douglas C.
    [J]. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2006, 317 (03): : 1027 - 1035