Discovery and structure-activity relationship of pyrrolo[2,1-f][1,2,4]triazines as inhibitors of phosphatidylinositol 3-kinase δ (PI3Kδ) for the treatment of immunological disorders

被引:0
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作者
Shi, Qing [1 ]
Marcoux, David [1 ]
Liu, Qingjie [1 ]
Batt, Douglas [1 ]
Cornelius, Lyndon [1 ]
Srivastava, Anurag [1 ]
Cherney, Robert [1 ]
Qin, Lan-ying [1 ]
Ruan, Zheming [1 ]
Neels, James [1 ]
Bhide, Rajeev [1 ]
Li, Ling [1 ]
Bertrand, Myra Beaudoin [1 ]
Gong, Hua [1 ]
Watterson, Scott [1 ]
Pan, Jie [1 ]
Tang, Huaping [1 ]
Fan, Jingsong [1 ]
Yarde, Melissa [1 ]
Cvijic, Mary Ellen [1 ]
Obermeier, Mary [1 ]
Fura, Aberra [1 ]
Weigelt, Carolyn [1 ]
Galella, Michael [1 ]
Sack, Jack [1 ]
Muckelbauer, Jodi [1 ]
Gillooly, Kathleen [1 ]
McIntyre, Kim [1 ]
Ruan, Qian [1 ]
Poss, Michael [1 ]
Hynes, John [1 ]
Macor, John [1 ]
Carter, Percy [1 ]
Ruepp, Stefan [1 ]
Schieven, Gary [1 ]
Tino, Joseph [1 ]
机构
[1] Bristol Myers Squibb, Princeton, NJ USA
关键词
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
36
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页数:1
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