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- [1] Discovery and SAR of pyrrolo[2,1-f][1,2,4]triazin-4-amines as potent and selective PI3Kδ inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (17) : 4256 - 4260Bhide, Rajeev S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USANeels, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAQin, Lan-Ying论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USARuan, Zheming论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAStachura, Sylwia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAWeigelt, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Mol Struct & Design, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USASack, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Mol Struct & Design, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAStefanski, Kevin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, PCO Discovery, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAGu, Xiaomei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, PCO Discovery, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAXie, Jenny H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAGoldstine, Christine B.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USASkala, Stacey论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAPedicord, Donna L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USARuepp, Stefan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, PCO Discovery, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USADhar, T. G. Murali论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USACarter, Percy H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USASalter-Cid, Luisa M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USAPoss, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USADavies, Paul论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08534 USA
- [2] Discovery and development of p38 MAP kinase inhibitors derived from pyrrolo[2,1-f][1,2,4]triazinesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U2722 - U2722Hynes, John, Jr.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USADyckman, Alaric论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USALi, Tianle论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USALin, Shuqun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAWrobleski, Stephen T.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USALoo, Derek论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAMcIntyre, Kim W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USASchieven, Gary L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAZhang, Rosemary论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAGillooly, Kathleen M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAPitt, Sidney论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAShen, Ding Ren论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USAShuster, David J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USADoweyko, Arthur论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USASack, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USABarrish, Joel C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USADodd, John H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USALeftheris, Katerina论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Pharmaceut Res Inst, Discovery Chem, Princeton, NJ 08543 USA
- [3] Discovery and Process Synthesis of Novel 2,7-Pyrrolo[2,1-f][1,2,4]triazinesORGANIC LETTERS, 2011, 13 (16) : 4204 - 4207Thieu, Tho论文数: 0 引用数: 0 h-index: 0机构: Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USASclafani, Joseph A.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Chem Proc Res & Dev, Worldwide Drug Dev, Malvern, PA 19355 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USALevy, Daniel V.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Chem Proc Res & Dev, Worldwide Drug Dev, Malvern, PA 19355 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USAMcLean, Andrew论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Chem Proc Res & Dev, Worldwide Drug Dev, Malvern, PA 19355 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USABreslin, Henry J.论文数: 0 引用数: 0 h-index: 0机构: Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USAOtt, Gregory R.论文数: 0 引用数: 0 h-index: 0机构: Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USABakale, Roger P.论文数: 0 引用数: 0 h-index: 0机构: Cephalon Inc, Chem Proc Res & Dev, Worldwide Drug Dev, Malvern, PA 19355 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USADorsey, Bruce D.论文数: 0 引用数: 0 h-index: 0机构: Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USA Worldwide Discovery Res, Dept Med Chem, W Chester, PA 19380 USA
- [4] Efficient, Scalable Synthesis of Functionalized Pyrrolo[2,1-f][1,2,4]triazinesORGANIC PROCESS RESEARCH & DEVELOPMENT, 2024, 28 (07) : 2765 - 2769Pack, Shawn K.论文数: 0 引用数: 0 h-index: 0机构: Kinnate Biopharm Inc, CMC, San Diego, CA 92130 USA Kinnate Biopharm Inc, CMC, San Diego, CA 92130 USAFeng, Lei论文数: 0 引用数: 0 h-index: 0机构: Pharmaron, Discovery Proc Chem, Xian 710018, Shaanxi, Peoples R China Kinnate Biopharm Inc, CMC, San Diego, CA 92130 USAChen, Ce论文数: 0 引用数: 0 h-index: 0机构: Pharmaron, Discovery Proc Chem, Xian 710018, Shaanxi, Peoples R China Kinnate Biopharm Inc, CMC, San Diego, CA 92130 USALi, Zhongzhen论文数: 0 引用数: 0 h-index: 0机构: Pharmaron, Discovery Proc Chem, Xian 710018, Shaanxi, Peoples R China Kinnate Biopharm Inc, CMC, San Diego, CA 92130 USA
- [5] Synthesis and SAR of new pyrrolo[2,1-f][1,2,4] triazines as potent p38α MAP kinase inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (08) : 2739 - 2744Wrobleski, Stephen T.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USALin, Shuqun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAHynes, John, Jr.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAWu, Hong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAPitt, Sidney论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAShen, Ding Ren论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAZhang, Rosemary论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAGillooly, Kathleen M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAShuster, David J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAMcIntyre, Kim W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USADoweyko, Arthur M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Struct Biol & Modeling, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAKish, Kevin F.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Struct Biol & Modeling, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USATredup, Rey A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Struct Biol & Modeling, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USADuke, Gerald J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Struct Biol & Modeling, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USASack, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Struct Biol & Modeling, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USAMcKinnon, Murray论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USADodd, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USABarrish, Joel C.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USASchieven, Gary L.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Immunol Drug Discovery, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USALeftheris, Katerina论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Dept Chem Immunol, Princeton, NJ 08543 USA
- [6] Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 27 (04) : 855 - 861Qin, Lan-Ying论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USARuan, Zheming论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USACherney, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USADhar, T. G. Murali论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USANeels, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAWeigelt, Carolyn A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USASack, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USASrivastava, Anurag S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USACornelius, Lyndon A. M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USATino, Joseph A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAStefanski, Kevin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAGu, Xiaomei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAXie, Jenny论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USASusulic, Vojkan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAYang, Xiaoxia论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAYarde-Chinn, Melissa论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USASkala, Stacey论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USABosnius, Ruth论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAGoldstein, Christine论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USADavies, Paul论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USARuepp, Stefan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USASalter-Cid, Luisa论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USABhide, Rajeev S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USAPoss, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA Bristol Myers Squibb, Rt 206 & Prov Line Rd, Princeton, NJ 08540 USA
- [7] Discovery of the pyrrolo[2,1-f][1,2,4]triazine nucleus as a new kinase inhibitor templateJOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (16) : 4054 - 4059Hunt, JT论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAMitt, T论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USABorzilleri, R论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAGullo-Brown, J论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAFargnoli, J论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAFink, B论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAHan, WC论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAMortillo, S论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAVite, G论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAWautlet, B论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAWong, T论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAYu, CA论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USAZheng, XP论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USABhide, R论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Pharmaceut Res Inst, Dept Oncol Chem, Princeton, NJ 08543 USA
- [8] Identification of pyrrolo[2,1-f][1,2,4] triazine-based inhibitors of Met kinaseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (06) : 1945 - 1951Schroeder, Gretchen M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAChen, Xiao-Tao论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAWilliams, David K.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USANirschl, David S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USACai, Zhen-Wei论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAWei, Donna论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USATokarski, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAAn, Yongmi论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USASack, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAChen, Zhong论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAHuynh, Tram论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAVaccaro, Wayne论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAPoss, Michael论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAWautlet, Barri论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAGullo-Brown, Johnni论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAKellar, Kristen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAManne, Veeraswamy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAHunt, John T.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAWong, Tai W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USALombardo, Louis J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USAFargnoli, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USABorzilleri, Robert M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA Bristol Myers Squibb Res & Dev, Princeton, NJ 08543 USA
- [9] Discovery of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of adaptor protein 2-associated kinase 1 for the treatment of painMEDICINAL CHEMISTRY RESEARCH, 2023, 32 (07) : 1369 - 1375Dzierba, Carolyn D. D.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USADasgupta, Bireshwar论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Neurosci Chem, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAKarageorge, George论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Neurosci Chem, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAKostich, Walter论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Neurosci Biol, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAHamman, Brian论文数: 0 引用数: 0 h-index: 0机构: Lexicon Pharmaceut, 8800 Technol Forest Pl, The Woodlands, TX 77381 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAAllen, Jason论文数: 0 引用数: 0 h-index: 0机构: Lexicon Pharmaceut, 8800 Technol Forest Pl, The Woodlands, TX 77381 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAEsposito, Kim M. M.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Leads Discovery & Optimizat, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAPadmanabha, Ramesh论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb, Dept Leads Discovery & Optimizat, Res & Dev, POB 5400, Princeton, NJ 08543 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAGrace, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Pharmaceut Candidate Optimizat, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USALentz, Kimberley论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Pharmaceut Candidate Optimizat, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAMorrison, John论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Pharmaceut Candidate Optimizat, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAMorgan, Daniel论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Pharmaceut Candidate Optimizat, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USAEaston, Amy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Neurosci Biol, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USABourin, Clotilde论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Bristol Myers Squibb, Dept Neurosci Biol, Res & Dev, 5 Res Pkwy, Wallingford, CT 06492 USA Bristol Myers Squibb, Small Mol Drug Discovery, Res & Dev, 250 Water St, Cambridge, MA 02141 USABrowning, Marc R. 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- [10] Discovery of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of adaptor protein 2-associated kinase 1 for the treatment of painMedicinal Chemistry Research, 2023, 32 : 1369 - 1375Carolyn D. Dzierba论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryBireshwar Dasgupta论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryGeorge Karageorge论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryWalter Kostich论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryBrian Hamman论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJason Allen论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryKim M. Esposito论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryRamesh Padmanabha论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJames Grace论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryKimberley Lentz论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJohn Morrison论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryDaniel Morgan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryAmy Easton论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryClotilde Bourin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryMarc R. Browning论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryRamkumar Rajamani论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryAndrew Good论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryDawn D. Parker论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJodi K. Muckelbauer论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJaved Khan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryDaniel Camac论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryKaushik Ghosh论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryVivek Halan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJonathan S. Lippy论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryKenneth S. Santone论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryR. Rex Denton论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryRyan Westphal论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryLinda J. Bristow论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryCharles M. Conway论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJoanne J. Bronson论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug DiscoveryJohn E. Macor论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb,Small Molecule Drug Discovery