Synthesis and antimicrobial activities of phenanthryl and biphenyl chalcone derivatives

被引：0
|
作者：
Al-Issa, SA [1 ]
Ghulikah, HA [1 ]
机构：
[1] Girls Coll Educ, Dept Chem, Riyadh 11593, Saudi Arabia
来源：
ASIAN JOURNAL OF CHEMISTRY | 2003年 / 15卷 / 02期
关键词：
synthesis; antimicrobial activity; phenanthryl; biphenyl chalcones;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Reaction of 1,3-diaryl-2-propen-1-ones 1 with hydrazine hydrate and phenyl hydrazine produced different substituted 2-pyrazolines of the type 3 and 4; acetylation of 3 gave 5; treatment of 3 with benzoyl chloride and benzene sulphonyl chloride afforded compounds 6 and 7 respectively. Interaction of 3 with phenylisocyanate and phenylisothiocyanate gave 8 and 9 respectively. The antibacterial activity of some of these prepared derivatives was studied.
引用
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页码：583 / 590
页数：8
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