Easy access to β-halo amino esters and aziridine 2-carboxylic esters from halohydrins

被引：18
|
作者：
Boukhris, S [1 ]
Souizi, A [1 ]
机构：
[1] Univ Ibn Tofail, Lab Synth Organ & Agrochim, Dept Chim, Fac Sci, Kenitra, Morocco
来源：
TETRAHEDRON LETTERS | 2003年 / 44卷 / 16期
关键词：
D O I：
10.1016/S0040-4039(03)00631-2
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The halohydrins prepared from epoxide esters, were treated with hydroxylamine derivatives. In subsequent reaction with NaOH/K2CO3/Bu4NHSO4 the N-protected beta-halo alpha-aminoesters thus obtained were converted into N-hydroxy ariridine 2-carboxylic esters in good yields. (C) 2003 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码：3259 / 3261
页数：3
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