Synthesis of alkyl 5-aryl-7-methyl-1,5-dihydrotetrazolo-[1,5-a]pyrimidine-6-carboxylates

被引：18
|
作者：
Gein, V. L. [1 ]
Vladimirov, I. N. [1 ]
Fedorova, O. V. [2 ]
Kurbatova, A. A. [1 ]
Nosova, N. V. [1 ]
Krylova, I. V. [1 ]
Vakhrin, M. I. [1 ]
机构：
[1] Perm State Pharmaceut Acad, Perm 614990, Russia
[2] Russian Acad Sci, Ural Div, Postovskii Inst Organ Synth, Ekaterinburg, Russia
来源：
RUSSIAN JOURNAL OF ORGANIC CHEMISTRY | 2010年 / 46卷 / 05期
关键词：
Dihydro; Aromatic Aldehyde; Acetoacetate; Metal Bath; Methyl Acetoacetate;
D O I：
10.1134/S1070428010050180
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Alkyl 5-aryl-7-methyl-1,5-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylates were obtained by melting acetoacetic acid esters with 5-aminotetrazole and aromatic aldehyde.
引用
收藏
页码：699 / 705
页数：7
相关论文
共 50 条
  • [21] Synthesis of N,N-dimethyl(diethyl)-7-aryl-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamides
    Gein, V. L.
    Zamaraeva, T. M.
    Zorina, A. A.
    Levandovskaya, E. B.
    Nosova, N. V.
    Vakhrin, M. I.
    RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2009, 45 (06) : 942 - 943
  • [22] Synthesis of (7-Aryl-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidin-6-yl)(phenyl)methanones
    Gein, V. L.
    Prudnikova, A. N.
    Kurbatova, A. A.
    Dmitriev, M. V.
    RUSSIAN JOURNAL OF ORGANIC CHEMISTRY, 2020, 56 (03) : 395 - 399
  • [23] Synthesis of (7-Aryl-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidin-6-yl)(phenyl)methanones
    V. L. Gein
    A. N. Prudnikova
    A. A. Kurbatova
    M. V. Dmitriev
    Russian Journal of Organic Chemistry, 2020, 56 : 395 - 399
  • [24] SYNTHESIS AND ANTIMICROBIAL ACTIVITY OF N,7-DIARYL-5-METHYL-4,7-DIHYDROTETRAZOLO[1,5-a] PYRIMIDINE-6-ARBOXAMIDES
    Gein, V. L.
    Zamaraeva, T. M.
    Kurbatova, A. A.
    Voronina, E. V.
    Vakhrin, M. I.
    PHARMACEUTICAL CHEMISTRY JOURNAL, 2010, 44 (07) : 366 - 369
  • [25] Synthesis and hypoglycemic activity of methyl-6-aryl(hetaryl)-5-(2-furanoyl)-3,6-dihydrotetrazolo[1,5-a]pyrimidine-4-carboxylates
    Gein, V. L.
    Zamaraeva, T. M.
    Mishunin, V. V.
    Kotegov, V. P.
    RUSSIAN JOURNAL OF GENERAL CHEMISTRY, 2016, 86 (02) : 286 - 290
  • [26] Synthesis and antimicrobial activity of n,7-diaryl-5-methyl-4,7-dihydrotetrazolo[1,5-a] pyrimidine-6-arboxamides
    V. L. Gein
    T. M. Zamaraeva
    A. A. Kurbatova
    E. V. Voronina
    M. I. Vakhrin
    Pharmaceutical Chemistry Journal, 2010, 44 : 366 - 369
  • [27] Synthesis and hypoglycemic activity of methyl-6-aryl(hetaryl)-5-(2-furanoyl)-3,6-dihydrotetrazolo[1,5-a]pyrimidine-4-carboxylates
    V. L. Gein
    T. M. Zamaraeva
    V. V. Mishunin
    V. P. Kotegov
    Russian Journal of General Chemistry, 2016, 86 : 286 - 290
  • [28] Solvent-free Synthesis of 5-methyl-7-aryl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylic esters Catalyzed by Sulfamic Acid
    Yao, Changsheng
    Lei, Song
    Wang, Cuihua
    Yu, Chenxia
    Tu, Shujiang
    JOURNAL OF HETEROCYCLIC CHEMISTRY, 2008, 45 (06) : 1609 - 1613
  • [29] Methyl 7-(4-bromophenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxylate
    Yao, Chang-Sheng
    Yu, Chen-Xia
    Lei, Song
    Tu, Shu-Jiang
    ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE, 2007, 63 : O3808 - U3011
  • [30] Synthesis of diethyl 6-aryl-3,6-dihydrotetrazolo-[1,5-a]pyrimidine-4,5-dicarboxylates
    V. L. Gein
    T. M. Zamaraeva
    M. V. Dmitriev
    Russian Journal of Organic Chemistry, 2016, 52 : 558 - 561
12345