Design and synthesis of cyclopropylamide analogs of combretastatin-A4 as novel microtubule-stabilizing agents

被引:0
|
作者
Li, Ke [1 ]
Chen, Huan [1 ]
Lv, Zhiliang [1 ]
Dong, Guoqiang [1 ]
Wang, Tiantian [1 ]
Liu, Jia [1 ]
Zhang, Mingfeng [1 ]
Li, Lingzhen [1 ]
Zhang, Tao [1 ]
Geng, Dongping [1 ]
Niu, Chunjuan [1 ]
Li, Yongmei [2 ]
机构
[1] Second Mil Med Univ, Dept Med Chem, Shanghai, Peoples R China
[2] Second Mil Med Univ, Changhai Hosp, Dept Oncol, Shanghai, Peoples R China
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2014年 / 247卷
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
325-MEDI
引用
收藏
页数:1
相关论文
共 50 条
  • [21] Molecular Mechanism of Action of Microtubule-Stabilizing Anticancer Agents
    Prota, Andrea E.
    Bargsten, Katja
    Zurwerra, Didier
    Field, Jessica J.
    Fernando Diaz, Jose
    Altmann, Karl-Heinz
    Steinmetz, Michel O.
    SCIENCE, 2013, 339 (6119) : 587 - 590
  • [22] Synthesis and pharmacological evaluation of combretastatin-A4 analogs of pyrazoline and pyridine derivatives as anticancer, anti-inflammatory and antioxidant agents
    Sadanand N. Shringare
    Hemant V. Chavan
    Pravin S. Bhale
    Sakharam B. Dongare
    Yoginath B. Mule
    Sandeep B. Patil
    Babasaheb P. Bandgar
    Medicinal Chemistry Research, 2018, 27 : 1226 - 1237
  • [23] Microtubule-stabilizing agents as potential therapeutics for neurodegenerative disease
    Brunden, Kurt R.
    Trojanowski, John Q.
    Smith, Amos B., III
    Lee, Virginia M. -Y.
    Ballatore, Carlo
    BIOORGANIC & MEDICINAL CHEMISTRY, 2014, 22 (18) : 5040 - 5049
  • [24] A SENSITIVE ASSAY FOR TAXOL AND OTHER MICROTUBULE-STABILIZING AGENTS
    SMITH, CD
    MOOBERRY, SL
    ZHANG, XQ
    HELT, AM
    CANCER LETTERS, 1994, 79 (02) : 213 - 219
  • [25] Synthesis and pharmacological evaluation of combretastatin-A4 analogs of pyrazoline and pyridine derivatives as anticancer, anti-inflammatory and antioxidant agents
    Shringare, Sadanand N.
    Chavan, Hemant V.
    Bhale, Pravin S.
    Dongare, Sakharam B.
    Mule, Yoginath B.
    Patil, Sandeep B.
    Bandgar, Babasaheb P.
    MEDICINAL CHEMISTRY RESEARCH, 2018, 27 (04) : 1226 - 1237
  • [26] Efficient synthesis and cytotoxicity of novel microtubule-stabilizing agent ceratamine A analogues
    Tao, Lulu
    Pan, Xuan
    Ji, Ming
    Chen, Xiaoguang
    Liu, Zhanzhu
    TETRAHEDRON, 2017, 73 (15) : 2159 - 2171
  • [27] Total synthesis of microtubule-stabilizing agent (-)-laulimalide
    Ghosh, AK
    Wang, Y
    Kim, JT
    JOURNAL OF ORGANIC CHEMISTRY, 2001, 66 (26): : 8973 - 8982
  • [28] Total synthesis of the microtubule-stabilizing agent (-)-laulimalide
    Paterson, I
    De Savi, C
    Tudge, M
    ORGANIC LETTERS, 2001, 3 (20) : 3149 - 3152
  • [29] Total Synthesis of Microtubule-Stabilizing Agent Ceratamine A
    Feng, Qiguo
    Tao, Lulu
    Liu, Zhanzhu
    JOURNAL OF ORGANIC CHEMISTRY, 2013, 78 (24): : 12814 - 12818
  • [30] Fighting cancer with microtubule-stabilizing agents: a computational investigation of the complex between β-tubulin and the microtubule-stabilizing, antitumor marine diterpenoid sarcodictyin A
    Pietra, Francesco
    STRUCTURAL CHEMISTRY, 2020, 31 (03) : 927 - 935