Histamine H1 receptor antagonist duration in recombinant receptor and isolated tissue assays

被引:0
|
作者
Browning, C. [1 ]
Nash, V. [1 ]
Russell, L. [1 ]
机构
[1] GlaxoSmithKline Inc, Stevenage, Herts, England
关键词
D O I
暂无
中图分类号
R392 [医学免疫学];
学科分类号
100102 ;
摘要
引用
收藏
页码:122 / 122
页数:1
相关论文
共 50 条
  • [31] Expression of histamine H1 receptor in placenta
    Matsuyama, K
    Kawakami, N
    Ichikawa, T
    Nitta, Y
    Ishimura, K
    Horio, S
    Fukui, H
    INFLAMMATION RESEARCH, 2004, 53 (Suppl 1) : S85 - S86
  • [32] HOMOLOGOUS HISTAMINE H1 RECEPTOR DESENSITIZATION RESULTS IN REDUCTION OF H1 RECEPTOR AGONIST EFFICACY
    LEURS, R
    SMIT, MJ
    BAST, A
    TIMMERMAN, H
    EUROPEAN JOURNAL OF PHARMACOLOGY, 1991, 196 (03) : 319 - 322
  • [33] Effects of Olopatadine Hydrochloride, a Histamine H1 Receptor Antagonist, on Histamine-Induced Skin Responses
    Hashimoto, Takashi
    Ishii, Norito
    Hamada, Takahiro
    Dainichi, Teruki
    Karashima, Tadashi
    Nakama, Takekuni
    Yasumoto, Shinichiro
    DERMATOLOGY RESEARCH AND PRACTICE, 2010, 2010
  • [34] BILASTINE Histamine H1 Receptor Antagonist Treatment of Allergic Rhinitis Treatment of Urticaria
    Ferrer, E.
    Pandian, R.
    Bolos, J.
    Castaner, R.
    DRUGS OF THE FUTURE, 2010, 35 (02) : 98 - 105
  • [35] Effect of Ions and Sequence Variants on the Antagonist Binding Properties of the Histamine H1 Receptor
    Conrad, Marcus
    Soeldner, Christian A.
    Sticht, Heinrich
    INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2022, 23 (03)
  • [36] In vivo pharmacological characterisation of bilastine, a potent and selective histamine H1 receptor antagonist
    Corcóstegui R.
    Labeaga L.
    Innerárity A.
    Berisa A.
    Orjales A.
    Drugs in R & D, 2006, 7 (4) : 219 - 231
  • [37] Pharmacological profile of histaprodifens at four recombinant histamine H1 receptor species isoforms
    Strasser, Andrea
    Striegl, Birgit
    Wittmann, Hans-Joachim
    Seifert, Roland
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2008, 324 (01): : 60 - 71
  • [38] Synthesis and Dual Histamine H1 and H2 Receptor Antagonist Activity of Cyanoguanidine Derivatives
    Sadek, Bassem
    Alisch, Rudi
    Buschauer, Armin
    Elz, Sigurd
    MOLECULES, 2013, 18 (11) : 14186 - 14202
  • [39] The histamine H1 receptor gene polymorphisms and schizophrenia
    Godlewska, B
    Limon, J
    Landowski, J
    AMERICAN JOURNAL OF MEDICAL GENETICS PART B-NEUROPSYCHIATRIC GENETICS, 2004, 130B (01): : 87 - 87
  • [40] LIGAND RECOGNITION MECHANISM OF THE HISTAMINE H1 RECEPTOR
    OHTA, K
    HAYASHI, H
    MIZUGUCHI, H
    KAGAMIYAMA, H
    FUJIMOTO, K
    FUKUI, H
    JOURNAL OF NEUROCHEMISTRY, 1995, 65 : S29 - S29