Functionalized Triarylsulfonium Salts for Aromatic [18F]Fluorination of Drug-like Small Molecules

被引：0
|
作者：
Sander, Kerstin [1 ]
Gendron, Thibault [1 ]
Yiannaki, Elena [2 ]
Cybulska, Klaudia [2 ]
Kalber, Tammy L. [3 ]
Lythgoe, Mark [3 ]
Arstad, Erik [1 ,2 ]
机构：
[1] UCL, Inst Nucl Med Radiochem, London, England
[2] UCL, Dept Chem, London, England
[3] UCL, Ctr Adv Biomed Imaging, London, England
来源：
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2015年 / 58卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学];
学科分类号：
071010 ; 081704 ;
摘要：
004
引用
收藏
页码：S4 / S4
页数：1
相关论文
共 50 条
  • [41] Automated synthesis of 18F radiolabelled indole containing Oncrasin-like molecules; a comparison of iodonium salts and boronic ester chemistry
    Alexander F. McDonald
    Yit Wooi Goh
    Jonathan M. White
    Andrew M. Scott
    Uwe Ackermann
    EJNMMI Radiopharmacy and Chemistry, 5
  • [42] Automated synthesis of 18F radiolabelled indole containing Oncrasin-like molecules; a comparison of iodonium salts and boronic ester chemistry
    McDonald, Alexander F.
    Goh, Yit Wooi
    White, Jonathan M.
    Scott, Andrew M.
    Ackermann, Uwe
    EJNMMI RADIOPHARMACY AND CHEMISTRY, 2020, 5 (01)
  • [43] Microwave-induced nucleophilic [18F]fluorination on aromatic rings:: Synthesis and effect of halogen on [18F]fluoride substitution of meta-halo (F, Cl, Br, I)-benzonitrile derivatives
    Guo, Ning
    Alagille, David
    Tamagnan, Gilles
    Price, Ronald R.
    Baldwin, Ronald M.
    APPLIED RADIATION AND ISOTOPES, 2008, 66 (10) : 1396 - 1402
  • [44] A machine-learning-assisted study of the permeability of small drug-like molecules across lipid membranes
    Chen, Guang
    Shen, Zhiqiang
    Li, Ying
    PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2020, 22 (35) : 19687 - 19696
  • [45] SYNTHESIS AND AROMATIC [F-18]FLUORINATION OF meta-POSITION ON PHENYL RING OF DONEPEZIL USING IODONIUM SALTS
    Jeon, Y. S.
    Moon, B. S.
    Kim, J. S.
    Kim, S. E.
    Lee, B. C.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2009, 52 : S212 - S212
  • [46] Synthesis of novel drug-like small molecules library based on IH-benzo[d]imidazcie
    Parmar, Tejasvi H.
    Sangani, Chetan B.
    Kulkarni, Mahesh
    AUSTRALIAN JOURNAL OF CHEMISTRY, 2022, 75 (04) : 276 - 284
  • [47] Novel drug-like small molecules protect from stress-induced gastric ulceration in vivo
    Kudryavtsev, K. V.
    Kucherenko, M. I.
    Falalyeyeva, T. M.
    Beregova, T. V.
    Ostapchenko, L. I.
    EUROPEAN JOURNAL OF CLINICAL INVESTIGATION, 2012, 42 : 6 - 6
  • [48] OPLS3: A Force Field Providing Broad Coverage of Drug-like Small Molecules and Proteins
    Harder, Edward
    Damm, Wolfgang
    Maple, Jon
    Wu, Chuanjie
    Reboul, Mark
    Xiang, Jin Yu
    Wang, Lingle
    Lupyan, Dmitry
    Dahlgren, Markus K.
    Knight, Jennifer L.
    Kaus, Joseph W.
    Cerutti, David S.
    Krilov, Goran
    Jorgensen, William L.
    Abel, Robert
    Friesner, Richard A.
    JOURNAL OF CHEMICAL THEORY AND COMPUTATION, 2016, 12 (01) : 281 - 296
  • [49] Ring-Closing Synthesis of Dibenzothiophene Sulfonium Salts and Their Use as Leaving Groups for Aromatic 18F-Fluorination
    Gendron, Thibault
    Sander, Kerstin
    Cybulska, Klaudia
    Benhamou, Laure
    Sin, Pak Kwan Brian
    Khan, Aqsa
    Wood, Michael
    Porter, Michael J.
    Arstad, Erik
    JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2018, 140 (35) : 11125 - 11132
  • [50] A Versatile Isocyanate-Mediated Strategy for Appending Chemical Tags onto Drug-Like Small Molecules
    Henry, Catherine C.
    Kruell, Jasmin A.
    Wilson, Robert M.
    Chang, Chia-Fu
    Woo, Christina M.
    Koehler, Angela N.
    BIOCONJUGATE CHEMISTRY, 2023, 34 (12) : 2181 - 2186
12345