Functionalized Triarylsulfonium Salts for Aromatic [18F]Fluorination of Drug-like Small Molecules

被引：0
|
作者：
Sander, Kerstin [1 ]
Gendron, Thibault [1 ]
Yiannaki, Elena [2 ]
Cybulska, Klaudia [2 ]
Kalber, Tammy L. [3 ]
Lythgoe, Mark [3 ]
Arstad, Erik [1 ,2 ]
机构：
[1] UCL, Inst Nucl Med Radiochem, London, England
[2] UCL, Dept Chem, London, England
[3] UCL, Ctr Adv Biomed Imaging, London, England
来源：
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2015年 / 58卷
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学];
学科分类号：
071010 ; 081704 ;
摘要：
004
引用
收藏
页码：S4 / S4
页数：1
相关论文
共 50 条
  • [1] Sulfonium Salts as Leaving Groups for Aromatic Labelling of Drug-like Small Molecules with Fluorine-18
    Kerstin Sander
    Thibault Gendron
    Elena Yiannaki
    Klaudia Cybulska
    Tammy L. Kalber
    Mark F. Lythgoe
    Erik Årstad
    Scientific Reports, 5
  • [2] Sulfonium Salts as Leaving Groups for Aromatic Labelling of Drug-like Small Molecules with Fluorine-18
    Sander, Kerstin
    Gendron, Thibault
    Yiannaki, Elena
    Cybulska, Klaudia
    Kalber, Tammy L.
    Lythgoe, Mark F.
    Arstad, Erika
    SCIENTIFIC REPORTS, 2015, 5
  • [3] 18F-Radiolabeling of Aromatic Compounds Using Triarylsulfonium Salts
    Mu, Linjing
    Fischer, Cindy R.
    Holland, Jason P.
    Becaud, Jessica
    Schubiger, P. August
    Schibli, Roger
    Ametamey, Simon M.
    Graham, Keith
    Stellfeld, Timo
    Dinkelborg, Ludger M.
    Lehmann, Lutz
    EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, 2012, 2012 (05) : 889 - 892
  • [4] Efficient automated production of [18F]flumazenil through aromatic fluorination of an iodonium salts precursor
    Moon, Byung Seok
    Park, Jun Hyung
    Lee, Hong Jin
    Kil, Hee Sup
    Chi, Dae Yoon
    Lee, Byung Chul
    Kim, Yu Kyeong
    Kim, Sang Eun
    JOURNAL OF NUCLEAR MEDICINE, 2010, 51
  • [5] 18F-labeling of unactivated aromatic compounds using triarylsulfonium salts
    Fischer, C.
    Mu, L.
    Becaud, J.
    Schubiger, P. A.
    Schibli, R.
    Ametamey, S. M.
    Graham, K.
    Stellfeld, T.
    Dinkelborg, L. M.
    Lehmann, L.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2011, 54 : S71 - S71
  • [6] Cu-catalyzed selective [18F]fluorination of (mesityl)(aryl)iodonium salts with K[18F]F
    Ichiishi, Naoko
    Brooks, Allen F.
    Topscewski, Joseph J.
    Rodnick, Melissa
    Sanford, Melanie S.
    Scott, Peter J. H.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248
  • [7] Copper-catalyzed [18F] fluorination of unsymmetrical diaryliodonium salts
    Ichiishi, Naoko
    Rodnick, Melissa
    Brooks, Allen
    Topczewski, Joseph
    Scott, Peter
    Sanford, Melanie
    JOURNAL OF NUCLEAR MEDICINE, 2014, 55
  • [8] Principles for targeting RNA with drug-like small molecules
    Katherine Deigan Warner
    Christine E. Hajdin
    Kevin M. Weeks
    Nature Reviews Drug Discovery, 2018, 17 : 547 - 558
  • [9] Principles for targeting RNA with drug-like small molecules
    Warner, Katherine Deigan
    Hajdin, Christine E.
    Weeks, Kevin M.
    NATURE REVIEWS DRUG DISCOVERY, 2018, 17 (08) : 547 - 558
  • [10] Site-Selective Late-Stage Aromatic [18F]Fluorination via Aryl Sulfonium Salts
    Xu, Peng
    Zhao, Da
    Berger, Florian
    Hamad, Aboubakr
    Rickmeier, Jens
    Petzold, Roland
    Kondratiuk, Mykhailo
    Bohdan, Kostiantyn
    Ritter, Tobias
    ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2020, 59 (05) : 1956 - 1960
12345