EVALUATION OF THE NK1 RECEPTOR ANTAGONIST SERLOPITANT IN PATIENTS WITH OVERACTIVE BLADDER

被引：0
|
作者：
Frenkl, Tara L.
Seltzer, Olga
Zhu, Haiyuan
Reiss, Theodore F.
Green, Stuart A.
Green, Stuart A.
机构：
来源：
JOURNAL OF UROLOGY | 2009年 / 181卷 / 04期
关键词：
D O I：
10.1016/S0022-5347(09)61895-4
中图分类号：
R5 [内科学]; R69 [泌尿科学（泌尿生殖系疾病）];
学科分类号：
1002 ; 100201 ;
摘要：
1873
引用
收藏
页码：676 / 676
页数：1
相关论文
共 50 条
  • [31] Synthesis of a tetrahydropyran NK1 receptor antagonist via asymmetric conjugate addition
    Huffman, MA
    Smitrovich, JH
    Rosen, JD
    Boice, GN
    Qu, CX
    Nelson, TD
    McNamara, JM
    JOURNAL OF ORGANIC CHEMISTRY, 2005, 70 (11): : 4409 - 4413
  • [32] Efficacy benefit of an NK1 receptor antagonist (NK1RA) in patients receiving carboplatin: supportive evidence with NEPA (a fixed combination of the NK1 RA, netupitant, and palonosetron) and aprepitant regimens
    Jordan, Karin
    Gralla, Richard
    Rizzi, Giada
    Kashef, Kimia
    SUPPORTIVE CARE IN CANCER, 2016, 24 (11) : 4617 - 4625
  • [33] Efficacy benefit of an NK1 receptor antagonist (NK1RA) in patients receiving carboplatin: supportive evidence with NEPA (a fixed combination of the NK1 RA, netupitant, and palonosetron) and aprepitant regimens
    Karin Jordan
    Richard Gralla
    Giada Rizzi
    Kimia Kashef
    Supportive Care in Cancer, 2016, 24 : 4617 - 4625
  • [34] The involvement of the NK1 receptor in neutrophil accumulation:: A study in wildtype and NK1 receptor knockout mice
    Cao, T
    Pinter, E
    Al-Rashed, S
    Gerard, NP
    Brain, SD
    BRITISH JOURNAL OF PHARMACOLOGY, 2000, 129 : U55 - U55
  • [35] Evaluation of selective NK1 receptor antagonist CI-1021 in animal models of inflammatory and neuropathic pain
    Gonzalez, MI
    Field, MJ
    Hughes, J
    Singh, L
    JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 2000, 294 (02): : 444 - 450
  • [36] Effect of an NK1/NK2 receptor antagonist on airway responses and inflammation to allergen in asthma
    Boot, Johan D.
    de Haas, Sanne
    Tarasevych, Svetlana
    Roy, Christine
    Wang, Lin
    Amin, Dilip
    Cohen, Judith
    Sterk, Peter J.
    Miller, Barry
    Paccaly, Anne
    Burggraaf, Jacobus
    Cohen, Adam F.
    Diamant, Zuzana
    AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2007, 175 (05) : 450 - 457
  • [37] NETUPITANT, A POTENT AND HIGHLY SELECTIVE NK1 RECEPTOR ANTAGONIST IN THE GUINEA-PIG ISOLATED URINARY BLADDER: COMPARISON WITH APREPITANT
    Palea, S.
    Rekik, M.
    Pietra, C.
    Lovati, E.
    Lluel, P.
    NEUROUROLOGY AND URODYNAMICS, 2010, 29 (06) : 992 - 994
  • [38] NETUPITANT, A POTENT AND HIGHLY SELECTIVE NK1 RECEPTOR ANTAGONIST IN THE GUINEA-PIG ISOLATED URINARY BLADDER: COMPARISON WITH APREPITANT
    Palea, S.
    Rekik, M.
    Pietra, C.
    Lovati, E.
    Lluel, P.
    INTERNATIONAL UROGYNECOLOGY JOURNAL, 2010, 21 : S188 - S190
  • [39] In vitro and in vivo pharmacological characterization of the novel NK1 receptor selective antagonist Netupitant
    Rizzi, Anna
    Campi, Barbara
    Camarda, Valeria
    Molinari, Stefano
    Cantoreggi, Sergio
    Regoli, Domenico
    Pietra, Claudio
    Calo, Girolamo
    PEPTIDES, 2012, 37 (01) : 86 - 97
  • [40] Utilization of an intramolecular hydrogen bond to increase the CNS penetration of an NK1 receptor antagonist
    Ashwood, VA
    Field, MJ
    Horwell, DC
    Julien-Larose, C
    Lewthwaite, RA
    McCleary, S
    Pritchard, MC
    Raphy, J
    Singh, L
    JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44 (14) : 2276 - 2285
12345