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- [21] CYCLIZATION OF ETHYL (E)/(Z)-[2-(1-CYCLOHEXEN-1-YL)CYCLOHEXYLIDENE]CYANOACETATE TO 10-AMINO-1,2,3,4,5,6,7,8-OCTAHYDROPHENANTHRENE-9-CARBOXYLIC ACID - A ROUTE TO 1,2,3,4,5,6,7,8-OCTAHYDROPHENANTHRENE DERIVATIVESLIEBIGS ANNALEN, 1995, (08): : 1567 - 1570WILAMOWSKI, JKRASODOMSKI, WNOWAK, BSEPIOL, JJ
- [22] Design, Synthesis, and Biological Evaluation of 3-[4-(2-Hydroxyethyl)piperazin-1-yl]-7-(6-methoxypyridin-3-yl)-1-(2-propoxyethyl)pyrido[3,4-b]pyrazin-2(1H)-one, a Potent, Orally Active, Brain Penetrant Inhibitor of Phosphodiesterase 5 (PDE5)JOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (06) : 2656 - 2660Hughes, Robert O.Rogier, D. JosephJacobsen, E. JonWalker, John K.MacInnes, AlanBond, Brian R.Zhang, Lena L.Yu, YingZheng, YiRumsey, Jeanne M.Walgren, Jennie L.Curtiss, Sandra W.Fobian, Yvette M.Heasley, Steven E.Cubbage, Jerry W.Moon, Joseph B.Brown, David L.Acker, Brad A.Maddux, Todd M.Tollefson, Mike B.Mischke, Brent V.Owen, Dafydd R.Freskos, John N.Molyneaux, John M.Benson, Alan G.Blevis-Bal, Rhadika M.
- [23] Stereoselective synthesis of (2S,7S)-7-(4-phenoxymethyl)2-(1-N-hydroxyureidyl-3-butyn-4-yl)oxepane:: a potential anti-asthmatic drug candidateTETRAHEDRON-ASYMMETRY, 2005, 16 (05) : 935 - 939Gurjar, MKRao, BVKrishna, LMChorghade, MSLey, SV
- [24] Synthesis and biological characterization of novel hybrid 7-{[2-(4-phenyl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-2-ol and their heterocyclic bioisosteric analogues for dopamine D2 and D3 receptorsBIOORGANIC & MEDICINAL CHEMISTRY, 2004, 12 (16) : 4361 - 4373Dutta, AKVenkataraman, SKFei, XSKolhatkar, RZhang, SJReith, MEA
- [25] Identification of (S)-1-(2-(2,4-difluorophenyl)-4-oxothiazolidin-3-yl)-3-(4-((7-(3-(4-ethylpiperazin-1-yl)propoxy)-6-methoxyquinolin-4-yl) oxy)-3,5-difluorophenyl)urea as a potential anti-colorectal cancer agentEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2022, 239Qi, BaohuiWang, FeiHe, HuanFan, MengmengHu, LipingXiong, LiGong, GuoweiShi, ShengminSong, Xiaomeng
- [26] Direct C7 Functionalization of Tryptophan. Synthesis of Methyl (S)-2-((tert-Butoxycarbonyl) amino)-3-(7-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indol-3-yl)propanoateORGANIC SYNTHESES, 2015, 92 : 373 - +Amaike, KazumaLoach, Richard P.Movassaghi, Mohammad
- [27] ASYMMETRIC-SYNTHESIS AND PROPERTIES OF THE ENANTIOMERS OF THE ANTIBACTERIAL AGENT 7-(3-AMINOPYRROLIDIN-1-YL)-1-(2,4-DIFLUOROPHENYL)-1,4-DIHYDRO-6-FLUORO-4-OXO-1,8-NAPHTHYRIDINE-3-CARBOXYLIC ACID HYDROCHLORIDEJOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (08) : 1586 - 1590ROSEN, TCHU, DTWLICO, IMFERNANDES, PBSHEN, LBORODKIN, SPERNET, AG
- [28] Modification of agonist binding moiety in hybrid derivative 5/7-{[2-(4-aryl-piperazin-1-yl)-ethyl]-propyl-amino}-5,6,7,8-tetrahydro-naphthalen-1-ol/-2-amino versions: Impact on functional activity and selectivity for dopamine D2/D3 receptorsBIOORGANIC & MEDICINAL CHEMISTRY, 2013, 21 (11) : 3164 - 3174Gopishetty, BhaskarZhang, SuhongKharkar, Prashant S.Antonio, TamaraReith, MaartenDutta, Aloke K.
- [29] SYNTHESIS OF 7-(4'-FLUORO-3,3',5-TRIMETHYL[1,1'-BIPHENYL]-2-YL)-3-HYDROXY-5-OXO-5-C-13-HEPTANOIC ACID AND TRANS-6-[2-(4'-FLUORO-3,3',5-TRIMETHYL[1,1'-BIPHENYL]-2-YL)ETHYL]-3,4,5,6-TETRAHYDRO-6-C-13-4-HYDROXY-2H-PYRAN-2-ONEJOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 1987, 24 (07): : 839 - 849STOKKER, GE
- [30] Synthesis and Characterization of 2-(((2,7-Dihydroxynaphthalen-1-yl)methylene)amino)-3',6'-bis(ethylamino)-2',7'-dimethylspiro[isoindoline-1,9'-xanthen]-3-one and Colorimetric Detection of Uranium in WaterMOLBANK, 2023, 2023 (03)Mohammed, RahisaOgadi, PeaceSeth, Dennis M.Vibho, AmrutaaGallant, Sarah K.Waterman, Rory