Allosteric Modulators of G Protein-Coupled Receptors

被引:5
|
作者
Wells, Gregory J. [1 ]
机构
[1] Penn Drug Discovery Inst, Doylestown, PA 18902 USA
关键词
CHALLENGES; STRATEGIES; BIOSYNTHESIS; MARAVIROC; LIGANDS; SERIES; SAR;
D O I
10.2174/1568026614666140826115952
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
引用
收藏
页码:1735 / 1737
页数:3
相关论文
共 50 条
  • [31] Viral G protein-coupled receptors as modulators of cancer hallmarks
    van Senten, Jeffrey R.
    Fan, Tian Shu
    Siderius, Marco
    Smit, Martine J.
    PHARMACOLOGICAL RESEARCH, 2020, 156
  • [32] Strategies for the identification of allosteric modulators of G-protein-coupled receptors
    Burford, Neil T.
    Watson, John
    Bertekap, Robert
    Alt, Andrew
    BIOCHEMICAL PHARMACOLOGY, 2011, 81 (06) : 691 - 702
  • [33] Allosteric modulators of class B G-protein-coupled receptors
    Hoare, Sam R. J.
    CURRENT NEUROPHARMACOLOGY, 2007, 5 (03) : 168 - 179
  • [34] G protein-coupled receptors in atherosclerosis: cannabinoid receptors as novel modulators of atherogenesis
    Lanuti, M.
    Chiurchiu, V.
    FEBS JOURNAL, 2013, 280 : 408 - 408
  • [35] An allosteric modulator to control endogenous g protein-coupled receptors with light
    Gorostiza, P.
    JOURNAL OF NEUROCHEMISTRY, 2015, 134 : 62 - 62
  • [36] Structural Insights into Activation and Allosteric Modulation of G Protein-Coupled Receptors
    Kruse, Andrew C.
    MULTIFACETED ROLES OF CRYSTALLOGRAPHY IN MODERN DRUG DISCOVERY, 2015, : 19 - 26
  • [37] Allosteric modulation of G protein-coupled receptors: perspectives and recent developments
    Soudijn, W
    van Wijngaarden, I
    Ijzerman, AP
    DRUG DISCOVERY TODAY, 2004, 9 (17) : 752 - 758
  • [38] An allosteric modulator to control endogenous G protein-coupled receptors with light
    Pittolo, Ilvia
    Gomez-Santacana, Xavier
    Eckelt, Kay
    Rovira, Xavier
    Dalton, James
    Goudet, Cyril
    Pin, Jean-Philippe
    Llobet, Artur
    Giraldo, Jesus
    Llebaria, Amadeu
    Gorostiza, Pau
    NATURE CHEMICAL BIOLOGY, 2014, 10 (10) : 813 - +
  • [39] Dynamical Correlations Reveal Allosteric Sites in G Protein-Coupled Receptors
    Renault, Pedro
    Giraldo, Jesus
    INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 2021, 22 (01) : 1 - 21
  • [40] An allosteric modulator to control endogenous G protein-coupled receptors with light
    Silvia Pittolo
    Xavier Gómez-Santacana
    Kay Eckelt
    Xavier Rovira
    James Dalton
    Cyril Goudet
    Jean-Philippe Pin
    Artur Llobet
    Jesús Giraldo
    Amadeu Llebaria
    Pau Gorostiza
    Nature Chemical Biology, 2014, 10 : 813 - 815